BYL719 KINOMEscan - Dataset (ID:20263)
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Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Alpelisib | EGFR(L747-S752del, P753S) | 92.0 | 1000 | nM |
Alpelisib | MET | 92.0 | 100 | nM |
Alpelisib | KCC4 | 92.0 | 100 | nM |
Alpelisib | MARK1 | 92.0 | 1000 | nM |
Alpelisib | PIP5K1A | 92.0 | 100 | nM |
Alpelisib | DYRK1A | 92.0 | 100 | nM |
Alpelisib | ALK | 92.0 | 100 | nM |
Alpelisib | PIK4CB | 92.0 | 100 | nM |
Alpelisib | M4K1 | 92.0 | 100 | nM |
Alpelisib | FER | 92.0 | 1000 | nM |
Alpelisib | GRK4 | 92.0 | 100 | nM |
Alpelisib | KPCE | 92.0 | 100 | nM |
Alpelisib | ZAP70 | 92.0 | 100 | nM |
Alpelisib | WEE1 | 92.0 | 100 | nM |
Alpelisib | S6K1 | 92.0 | 100 | nM |
Alpelisib | MYO3A | 92.0 | 100 | nM |
Alpelisib | EPHB3 | 92.0 | 1000 | nM |
Alpelisib | EGFR(E746-A750del) | 93.0 | 1000 | nM |
Alpelisib | CAMK2A | 93.0 | 1000 | nM |
Alpelisib | CAMK2A | 93.0 | 100 | nM |
Alpelisib | NEK6 | 93.0 | 100 | nM |
Alpelisib | KIT(V559D,V654A) | 93.0 | 100 | nM |
Alpelisib | DAPK3 | 93.0 | 1000 | nM |
Alpelisib | AKT1 | 93.0 | 100 | nM |
Alpelisib | IKKE | 93.0 | 100 | nM |