BYL719 KINOMEscan - Dataset (ID:20263)

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Small Molecule Protein % Control Assay compound conc Conc unit
Alpelisib EGFR(L747-S752del, P753S) 92.0 1000
nM
Alpelisib MET 92.0 100
nM
Alpelisib KCC4 92.0 100
nM
Alpelisib MARK1 92.0 1000
nM
Alpelisib PIP5K1A 92.0 100
nM
Alpelisib DYRK1A 92.0 100
nM
Alpelisib ALK 92.0 100
nM
Alpelisib PIK4CB 92.0 100
nM
Alpelisib M4K1 92.0 100
nM
Alpelisib FER 92.0 1000
nM
Alpelisib GRK4 92.0 100
nM
Alpelisib KPCE 92.0 100
nM
Alpelisib ZAP70 92.0 100
nM
Alpelisib WEE1 92.0 100
nM
Alpelisib S6K1 92.0 100
nM
Alpelisib MYO3A 92.0 100
nM
Alpelisib EPHB3 92.0 1000
nM
Alpelisib EGFR(E746-A750del) 93.0 1000
nM
Alpelisib CAMK2A 93.0 1000
nM
Alpelisib CAMK2A 93.0 100
nM
Alpelisib NEK6 93.0 100
nM
Alpelisib KIT(V559D,V654A) 93.0 100
nM
Alpelisib DAPK3 93.0 1000
nM
Alpelisib AKT1 93.0 100
nM
Alpelisib IKKE 93.0 100
nM