BYL719 KINOMEscan - Dataset (ID:20263)

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Small Molecule Protein % Control Assay compound conc Conc unit
Alpelisib PKMYT1 90.0 1000
nM
Alpelisib PFCDPK1(P.falciparum) 90.0 1000
nM
Alpelisib LOK 90.0 1000
nM
Alpelisib PKAC-alpha 90.0 1000
nM
Alpelisib CDK4-cyclinD1 90.0 1000
nM
Alpelisib M3K5 90.0 1000
nM
Alpelisib AMPK-alpha1 91.0 1000
nM
Alpelisib MAP4K5 91.0 100
nM
Alpelisib TESK1 91.0 100
nM
Alpelisib ALK(L1196M) 91.0 100
nM
Alpelisib DYRK1A 91.0 1000
nM
Alpelisib DRAK1 91.0 100
nM
Alpelisib CAMK1D 91.0 1000
nM
Alpelisib SIK3 91.0 100
nM
Alpelisib IGF1R 91.0 100
nM
Alpelisib PAK4 91.0 1000
nM
Alpelisib FYN 91.0 100
nM
Alpelisib RET 91.0 1000
nM
Alpelisib CSNK1D 91.0 100
nM
Alpelisib RPS6KA5(Kin.Dom.2-C-terminal) 91.0 100
nM
Alpelisib PKN2 91.0 1000
nM
Alpelisib MK03 91.0 100
nM
Alpelisib AURKB 91.0 1000
nM
Alpelisib MELK 91.0 100
nM
Alpelisib EPHA6 91.0 1000
nM