BYL719 KINOMEscan - Dataset (ID:20263)

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Small Molecule Protein % Control Assay compound conc Conc unit
Alpelisib EPHA8 100.0 100
nM
Alpelisib CDK2 85.0 100
nM
Alpelisib EPHB1 99.0 100
nM
Alpelisib ACVR1 100.0 100
nM
Alpelisib EPHB2 98.0 100
nM
Alpelisib CDK3 100.0 100
nM
Alpelisib EPHB3 88.0 100
nM
Alpelisib M3K6 100.0 100
nM
Alpelisib EPHB4 81.0 100
nM
Alpelisib CDK4-cyclinD1 100.0 100
nM
Alpelisib EPHB6 100.0 100
nM
Alpelisib ABL1(F317L)-nonphosphorylated 98.0 100
nM
Alpelisib ERBB2 89.0 100
nM
Alpelisib CDK4-cyclinD1 89.0 100
nM
Alpelisib ERBB3 100.0 100
nM
Alpelisib AURKA 100.0 100
nM
Alpelisib ERBB4 100.0 100
nM
Alpelisib CDK4-cyclinD3 95.0 100
nM
Alpelisib MK03 91.0 100
nM
Alpelisib ACVR1B 100.0 100
nM
Alpelisib MK01 88.0 100
nM
Alpelisib CDK5 85.0 100
nM
Alpelisib ERK3 100.0 100
nM
Alpelisib AURKB 93.0 100
nM
Alpelisib OSR1 100.0 100
nM