BYL719 KINOMEscan - Dataset (ID:20263)
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Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Alpelisib | EPHA8 | 100.0 | 100 | nM |
Alpelisib | CDK2 | 85.0 | 100 | nM |
Alpelisib | EPHB1 | 99.0 | 100 | nM |
Alpelisib | ACVR1 | 100.0 | 100 | nM |
Alpelisib | EPHB2 | 98.0 | 100 | nM |
Alpelisib | CDK3 | 100.0 | 100 | nM |
Alpelisib | EPHB3 | 88.0 | 100 | nM |
Alpelisib | M3K6 | 100.0 | 100 | nM |
Alpelisib | EPHB4 | 81.0 | 100 | nM |
Alpelisib | CDK4-cyclinD1 | 100.0 | 100 | nM |
Alpelisib | EPHB6 | 100.0 | 100 | nM |
Alpelisib | ABL1(F317L)-nonphosphorylated | 98.0 | 100 | nM |
Alpelisib | ERBB2 | 89.0 | 100 | nM |
Alpelisib | CDK4-cyclinD1 | 89.0 | 100 | nM |
Alpelisib | ERBB3 | 100.0 | 100 | nM |
Alpelisib | AURKA | 100.0 | 100 | nM |
Alpelisib | ERBB4 | 100.0 | 100 | nM |
Alpelisib | CDK4-cyclinD3 | 95.0 | 100 | nM |
Alpelisib | MK03 | 91.0 | 100 | nM |
Alpelisib | ACVR1B | 100.0 | 100 | nM |
Alpelisib | MK01 | 88.0 | 100 | nM |
Alpelisib | CDK5 | 85.0 | 100 | nM |
Alpelisib | ERK3 | 100.0 | 100 | nM |
Alpelisib | AURKB | 93.0 | 100 | nM |
Alpelisib | OSR1 | 100.0 | 100 | nM |