BYL719 KINOMEscan - Dataset (ID:20263)
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Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Alpelisib | AMPK-alpha2 | 98.0 | 100 | nM |
Alpelisib | EGFR(L858R,T790M) | 94.0 | 100 | nM |
Alpelisib | CAMKK2 | 84.0 | 100 | nM |
Alpelisib | EGFR(L861Q) | 96.0 | 100 | nM |
Alpelisib | AAK1 | 79.0 | 100 | nM |
Alpelisib | EGFR(S752-I759del) | 100.0 | 100 | nM |
Alpelisib | CASK | 83.0 | 100 | nM |
Alpelisib | EGFR(T790M) | 100.0 | 100 | nM |
Alpelisib | ANKK1 | 100.0 | 100 | nM |
Alpelisib | EIF2AK1 | 98.0 | 100 | nM |
Alpelisib | CDC2L1 | 100.0 | 100 | nM |
Alpelisib | EPHA1 | 94.0 | 100 | nM |
Alpelisib | ABL2 | 93.0 | 100 | nM |
Alpelisib | EPHA2 | 93.0 | 100 | nM |
Alpelisib | CDC2L2 | 100.0 | 100 | nM |
Alpelisib | EPHA3 | 99.0 | 100 | nM |
Alpelisib | NUAK1 | 100.0 | 100 | nM |
Alpelisib | EPHA4 | 100.0 | 100 | nM |
Alpelisib | CDC2L5 | 98.0 | 100 | nM |
Alpelisib | EPHA5 | 81.0 | 100 | nM |
Alpelisib | ABL1(M351T)-phosphorylated | 100.0 | 100 | nM |
Alpelisib | EPHA6 | 89.0 | 100 | nM |
Alpelisib | CDK11 | 93.0 | 100 | nM |
Alpelisib | EPHA7 | 100.0 | 100 | nM |
Alpelisib | MST2 | 88.0 | 100 | nM |