BYL719 KINOMEscan - Dataset (ID:20263)

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Small Molecule Protein % Control Assay compound conc Conc unit
Alpelisib AMPK-alpha2 98.0 100
nM
Alpelisib EGFR(L858R,T790M) 94.0 100
nM
Alpelisib CAMKK2 84.0 100
nM
Alpelisib EGFR(L861Q) 96.0 100
nM
Alpelisib AAK1 79.0 100
nM
Alpelisib EGFR(S752-I759del) 100.0 100
nM
Alpelisib CASK 83.0 100
nM
Alpelisib EGFR(T790M) 100.0 100
nM
Alpelisib ANKK1 100.0 100
nM
Alpelisib EIF2AK1 98.0 100
nM
Alpelisib CDC2L1 100.0 100
nM
Alpelisib EPHA1 94.0 100
nM
Alpelisib ABL2 93.0 100
nM
Alpelisib EPHA2 93.0 100
nM
Alpelisib CDC2L2 100.0 100
nM
Alpelisib EPHA3 99.0 100
nM
Alpelisib NUAK1 100.0 100
nM
Alpelisib EPHA4 100.0 100
nM
Alpelisib CDC2L5 98.0 100
nM
Alpelisib EPHA5 81.0 100
nM
Alpelisib ABL1(M351T)-phosphorylated 100.0 100
nM
Alpelisib EPHA6 89.0 100
nM
Alpelisib CDK11 93.0 100
nM
Alpelisib EPHA7 100.0 100
nM
Alpelisib MST2 88.0 100
nM