BYL719 KINOMEscan - Dataset (ID:20263)

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Small Molecule Protein % Control Assay compound conc Conc unit
Alpelisib ABL1(Y253F)-phosphorylated 100.0 100
nM
Alpelisib ABL1(Y253F)-phosphorylated 100.0 1000
nM
Alpelisib ABL1(F317I)-phosphorylated 100.0 100
nM
Alpelisib AKT3 100.0 100
nM
Alpelisib ALK(L1196M) 100.0 1000
nM
Alpelisib AKT2 100.0 100
nM
Alpelisib AKT2 100.0 1000
nM
Alpelisib ABL1(M351T)-phosphorylated 100.0 100
nM
Alpelisib ACVR1 100.0 100
nM
Alpelisib ACVR1 100.0 1000
nM
Alpelisib ACVR1B 100.0 100
nM
Alpelisib AMPK-alpha2 100.0 1000
nM
Alpelisib AURKA 100.0 1000
nM
Alpelisib AXL 100.0 1000
nM
Alpelisib ALK(C1156Y) 100.0 100
nM
Alpelisib BMPR2 100.0 1000
nM
Alpelisib M3K6 100.0 1000
nM
Alpelisib ACVRL1 100.0 1000
nM
Alpelisib ABL1(Q252H)-phosphorylated 100.0 1000
nM
Alpelisib ABL1(F317L)-phosphorylated 100.0 100
nM
Alpelisib ADCK4 100.0 100
nM
Alpelisib ADCK4 100.0 1000
nM
Alpelisib ABL1(T315I)-nonphosphorylated 100.0 1000
nM
Alpelisib CDC2L2 100.0 1000
nM
Alpelisib CDC2L2 100.0 100
nM