BYL719 KINOMEscan - Dataset (ID:20263)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Alpelisib | ABL1(Y253F)-phosphorylated | 100.0 | 100 | nM |
Alpelisib | ABL1(Y253F)-phosphorylated | 100.0 | 1000 | nM |
Alpelisib | ABL1(F317I)-phosphorylated | 100.0 | 100 | nM |
Alpelisib | AKT3 | 100.0 | 100 | nM |
Alpelisib | ALK(L1196M) | 100.0 | 1000 | nM |
Alpelisib | AKT2 | 100.0 | 100 | nM |
Alpelisib | AKT2 | 100.0 | 1000 | nM |
Alpelisib | ABL1(M351T)-phosphorylated | 100.0 | 100 | nM |
Alpelisib | ACVR1 | 100.0 | 100 | nM |
Alpelisib | ACVR1 | 100.0 | 1000 | nM |
Alpelisib | ACVR1B | 100.0 | 100 | nM |
Alpelisib | AMPK-alpha2 | 100.0 | 1000 | nM |
Alpelisib | AURKA | 100.0 | 1000 | nM |
Alpelisib | AXL | 100.0 | 1000 | nM |
Alpelisib | ALK(C1156Y) | 100.0 | 100 | nM |
Alpelisib | BMPR2 | 100.0 | 1000 | nM |
Alpelisib | M3K6 | 100.0 | 1000 | nM |
Alpelisib | ACVRL1 | 100.0 | 1000 | nM |
Alpelisib | ABL1(Q252H)-phosphorylated | 100.0 | 1000 | nM |
Alpelisib | ABL1(F317L)-phosphorylated | 100.0 | 100 | nM |
Alpelisib | ADCK4 | 100.0 | 100 | nM |
Alpelisib | ADCK4 | 100.0 | 1000 | nM |
Alpelisib | ABL1(T315I)-nonphosphorylated | 100.0 | 1000 | nM |
Alpelisib | CDC2L2 | 100.0 | 1000 | nM |
Alpelisib | CDC2L2 | 100.0 | 100 | nM |