BYL719 KINOMEscan - Dataset (ID:20263)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
|---|---|---|---|---|
| Alpelisib | EGFR(L858R) | 100.0 | 1000 | nM |
| Alpelisib | KKCC1 | 99.0 | 1000 | nM |
| Alpelisib | EGFR(L858R,T790M) | 100.0 | 1000 | nM |
| Alpelisib | MLK1 | 100.0 | 1000 | nM |
| Alpelisib | EGFR(L861Q) | 82.0 | 1000 | nM |
| Alpelisib | CAMKK2 | 88.0 | 1000 | nM |
| Alpelisib | EGFR(S752-I759del) | 98.0 | 1000 | nM |
| Alpelisib | AMPK-alpha2 | 100.0 | 1000 | nM |
| Alpelisib | EGFR(T790M) | 100.0 | 1000 | nM |
| Alpelisib | CASK | 71.0 | 1000 | nM |
| Alpelisib | EIF2AK1 | 100.0 | 1000 | nM |
| Alpelisib | ABL1-phosphorylated | 10.0 | 1000 | nM |
| Alpelisib | EPHA1 | 81.0 | 1000 | nM |
| Alpelisib | CDC2L1 | 100.0 | 1000 | nM |
| Alpelisib | EPHA2 | 84.0 | 1000 | nM |
| Alpelisib | ANKK1 | 100.0 | 1000 | nM |
| Alpelisib | EPHA3 | 100.0 | 1000 | nM |
| Alpelisib | CDC2L2 | 100.0 | 1000 | nM |
| Alpelisib | EPHA4 | 100.0 | 1000 | nM |
| Alpelisib | ABL1(H396P)-phosphorylated | 2.9 | 1000 | nM |
| Alpelisib | EPHA5 | 100.0 | 1000 | nM |
| Alpelisib | CDC2L5 | 100.0 | 1000 | nM |
| Alpelisib | EPHA6 | 91.0 | 1000 | nM |
| Alpelisib | NUAK1 | 100.0 | 1000 | nM |
| Alpelisib | MST2 | 94.0 | 1000 | nM |