GDC-0941 KINOMEscan-3 - Dataset (ID:20261)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Pictilisib | PIK3CB | 15.0 | 100 | nM |
Pictilisib | PIK3C2G | 17.0 | 1000 | nM |
Pictilisib | PIK3CA(H1047L) | 17.0 | 100 | nM |
Pictilisib | PIK3C2B | 18.0 | 1000 | nM |
Pictilisib | JAK1(JH2domain-pseudokinase) | 18.0 | 1000 | nM |
Pictilisib | RSK2(Kin.Dom.2-C-terminal) | 48.0 | 100 | nM |
Pictilisib | PIK3CG | 48.0 | 100 | nM |
Pictilisib | PIP5K1C | 51.0 | 100 | nM |
Pictilisib | MYLK4 | 52.0 | 1000 | nM |
Pictilisib | VRK2 | 54.0 | 1000 | nM |
Pictilisib | CLK2 | 55.0 | 1000 | nM |
Pictilisib | CLK4 | 56.0 | 1000 | nM |
Pictilisib | EPHB6 | 57.0 | 1000 | nM |
Pictilisib | HASP | 59.0 | 1000 | nM |
Pictilisib | MK12 | 59.0 | 1000 | nM |
Pictilisib | CLK1 | 59.0 | 1000 | nM |
Pictilisib | FYV1 | 59.0 | 100 | nM |
Pictilisib | MKNK1 | 60.0 | 100 | nM |
Pictilisib | HIPK2 | 61.0 | 1000 | nM |
Pictilisib | FLT3(D835V) | 62.0 | 1000 | nM |
Pictilisib | CDC2L5 | 63.0 | 100 | nM |
Pictilisib | TNIK | 64.0 | 100 | nM |
Pictilisib | MLK3 | 64.0 | 100 | nM |
Pictilisib | EGFR(L747-S752del, P753S) | 64.0 | 100 | nM |
Pictilisib | KGP1 | 65.0 | 1000 | nM |