PF-3758309 KiNativ -- single dose experiment - Dataset (ID:20254)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| PF-3758309 | THP-1 | CRK7 | DIKCSNILLNNSGQIK | Lys2 | 8.2 | 1 | uM |
| PF-3758309 | THP-1 | ZC1/HGK,ZC2/TNIK,ZC3/MINK | DIKGQNVLLTENAEVK | Lys2 | 8.4 | 1 | uM |
| PF-3758309 | THP-1 | LKB1 | DIKPGNLLLTTGGTLK | Lys2 | 84.9 | 1 | uM |
| PF-3758309 | THP-1 | IRAK1 | AIQFLHQDSPSLIHGDIKSSNVLLDER | Lys2 | 8.6 | 1 | uM |
| PF-3758309 | THP-1 | IKKE,TBK1 | DIKPGNIMR | Lys2 | 87.6 | 1 | uM |
| PF-3758309 | THP-1 | IKKE | SGELVAVKVFNTTSYLRPR | Lys1 | 87.7 | 1 | uM |
| PF-3758309 | THP-1 | CDK4 | DLKPENILVTSGGTVK | Lys2 | -8.8 | 1 | uM |
| PF-3758309 | THP-1 | SRPK1/2 | FVAMKVVK | Lys1 | 89.2 | 1 | uM |
| PF-3758309 | THP-1 | CaMK2g | TSTQEYAAKIINTK | Lys1 | 89.3 | 1 | uM |
| PF-3758309 | THP-1 | MARK3 | EVAIKIIDKTQLNPTSLQK | Lys1 | 89.4 | 1 | uM |
| PF-3758309 | THP-1 | KCC2D | IPTGQEYAAKIINTK | Lys1 | 89.8 | 1 | uM |
| PF-3758309 | THP-1 | CDK2 | NKLTGEVVALKK | Lys1 | -9.0 | 1 | uM |
| PF-3758309 | THP-1 | MARK3,MARK4 | EVAIKIIDK | Lys1 | 90.1 | 1 | uM |
| PF-3758309 | THP-1 | MARK1,MARK2 | EVAVKIIDK | Lys1 | 90.2 | 1 | uM |
| PF-3758309 | THP-1 | RSK1,RSK2,RSK3_domain1 | DLKPENILLDEEGHIK | Lys2 | 90.6 | 1 | uM |
| PF-3758309 | THP-1 | INSR | VAVKTVNESASLR | Lys1 | 9.1 | 1 | uM |
| PF-3758309 | THP-1 | CHK2 | VAIKIISK | Lys1 | 91.1 | 1 | uM |
| PF-3758309 | THP-1 | DNAPK | EHPFLVKGGEDLR | ATP | 9.2 | 1 | uM |
| PF-3758309 | THP-1 | MAP3K1 | DVKGANLLIDSTGQR | Lys2 | -9.4 | 1 | uM |
| PF-3758309 | THP-1 | FRAP1 | IQSIAPSLQVITSKQRPR | ATP | 9.4 | 1 | uM |
| PF-3758309 | THP-1 | ULK1 | DLKPQNILLSNPAGR | Lys2 | -9.5 | 1 | uM |
| PF-3758309 | THP-1 | AMPKa1,AMPKa2 | DLKPENVLLDAHMNAK | Lys2 | 96.4 | 1 | uM |
| PF-3758309 | THP-1 | CDK7 | DLKPNNLLLDENGVLK | Lys2 | 96.5 | 1 | uM |
| PF-3758309 | THP-1 | AMPKa1,AMPKa2 | VAVKILNR | Lys1 | 97.6 | 1 | uM |