PF-3758309 KiNativ -- single dose experiment - Dataset (ID:20254)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| PF-3758309 | THP-1 | MK14 | QELNKTIWEVPER | Protein Kinase Domain | 7.4 | 1 | uM |
| PF-3758309 | THP-1 | CDK9 | DMKAANVLITR | Lys2 | -5.6 | 1 | uM |
| PF-3758309 | THP-1 | CDC2 | DLKPQNLLIDDKGTIK | Lys2 | -0.9 | 1 | uM |
| PF-3758309 | THP-1 | GSK3A | DIKPQNLLVDPDTAVLK | Lys2 | 52.6 | 1 | uM |
| PF-3758309 | THP-1 | IRAK1 | AIQFLHQDSPSLIHGDIKSSNVLLDER | Lys2 | 8.6 | 1 | uM |
| PF-3758309 | THP-1 | IRAK4 | DIKSANILLDEAFTAK | Lys2 | 4.0 | 1 | uM |
| PF-3758309 | THP-1 | CDK13 | DIKCSNILLNNR | Lys2 | -7.4 | 1 | uM |
| PF-3758309 | THP-1 | KC1G2 | DVKPENFLVGRPGTK | Lys2 | 7.7 | 1 | uM |
| PF-3758309 | THP-1 | MK01 | DLKPSNLLLNTTCDLK | Lys2 | 55.4 | 1 | uM |
| PF-3758309 | THP-1 | CaMK2a,CaMK2b,CaMK2d,CaMK2g | DLKPENLLLASK | Lys2 | 79.9 | 1 | uM |
| PF-3758309 | THP-1 | AMPKa1,AMPKa2 | DLKPENVLLDAHMNAK | Lys2 | 96.4 | 1 | uM |
| PF-3758309 | THP-1 | IKKE,TBK1 | DIKPGNIMR | Lys2 | 87.6 | 1 | uM |
| PF-3758309 | THP-1 | BRAF | DLKSNNIFLHEDLTVK | Lys2 | -5.4 | 1 | uM |
| PF-3758309 | THP-1 | CDK20 | DLKPANLLISASGQLK | Lys2 | 7.1 | 1 | uM |
| PF-3758309 | THP-1 | CRK7 | DIKCSNILLNNSGQIK | Lys2 | 8.2 | 1 | uM |
| PF-3758309 | THP-1 | CDK11,CDK8 | DLKPANILVMGEGPER | Lys2 | -29.4 | 1 | uM |
| PF-3758309 | THP-1 | CHK2 | DLKPENVLLSSQEEDCLIK | Lys2 | 81.8 | 1 | uM |
| PF-3758309 | THP-1 | CDK2 | DLKPQNLLINTEGAIK | Lys2 | 2.8 | 1 | uM |
| PF-3758309 | THP-1 | CDK4 | DLKPENILVTSGGTVK | Lys2 | -8.8 | 1 | uM |
| PF-3758309 | THP-1 | MK03 | DLKPSNLLINTTCDLK | Lys2 | 56.5 | 1 | uM |
| PF-3758309 | THP-1 | CDK5 | DLKPQNLLINR | Lys2 | -31.5 | 1 | uM |
| PF-3758309 | THP-1 | CDK6 | DLKPQNILVTSSGQIK | Lys2 | -6.4 | 1 | uM |
| PF-3758309 | THP-1 | CDK7 | DLKPNNLLLDENGVLK | Lys2 | 96.5 | 1 | uM |
| PF-3758309 | THP-1 | GSK3B | DIKPQNLLLDPDTAVLK | Lys2 | 74.7 | 1 | uM |
| PF-3758309 | THP-1 | LKB1 | DIKPGNLLLTTGGTLK | Lys2 | 84.9 | 1 | uM |