RAF-265 KINOMEscan - Dataset (ID:20201)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
RAF 265 | DDR1 | 13.0 | nM |
RAF 265 | EPHB6 | 43.0 | nM |
RAF 265 | YSK4 | 54.0 | nM |
RAF 265 | GCN2(Kin.Dom.2,S808G) | 55.0 | nM |
RAF 265 | LOK | 60.0 | nM |
RAF 265 | MLTK | 63.0 | nM |
RAF 265 | RET(M918T) | 72.0 | nM |
RAF 265 | KIT(L576P) | 83.0 | nM |
RAF 265 | CIT | 87.0 | nM |
RAF 265 | RET(V804M) | 89.0 | nM |
RAF 265 | TAOK2 | 140.0 | nM |
RAF 265 | TIE1 | 150.0 | nM |
RAF 265 | RET | 150.0 | nM |
RAF 265 | KIT(V559D) | 170.0 | nM |
RAF 265 | KIT | 200.0 | nM |
RAF 265 | PGFRB | 240.0 | nM |
RAF 265 | KIT(V559D,T670I) | 240.0 | nM |
RAF 265 | CSF1R | 250.0 | nM |
RAF 265 | ABL1-nonphosphorylated | 300.0 | nM |
RAF 265 | RET(V804L) | 320.0 | nM |
RAF 265 | BRAF(V600E) | 330.0 | nM |
RAF 265 | LYN | 370.0 | nM |
RAF 265 | RAF1 | 390.0 | nM |
RAF 265 | TYK2(JH1domain-catalytic) | 410.0 | nM |
RAF 265 | ABL1(Q252H)-nonphosphorylated | 440.0 | nM |