Dasatinib KINOMEscan - Dataset (ID:20196)

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Small Molecule Protein Kd Conc unit
Dasatinib EPHB2 0.39
nM
Dasatinib EPHB1 0.45
nM
Dasatinib PGFRA 0.47
nM
Dasatinib FGR 0.50
nM
Dasatinib KIT(L576P) 0.57
nM
Dasatinib LYN 0.57
nM
Dasatinib CSF1R 0.58
nM
Dasatinib PGFRB 0.63
nM
Dasatinib KIT(A829P) 0.66
nM
Dasatinib KIT(V559D) 0.68
nM
Dasatinib DDR1 0.69
nM
Dasatinib FYN 0.79
nM
Dasatinib KIT 0.81
nM
Dasatinib EPHA2 0.85
nM
Dasatinib CSK 1.00
nM
Dasatinib EPHA4 1.20
nM
Dasatinib BMX 1.40
nM
Dasatinib BTK 1.40
nM
Dasatinib KIT(D816H) 1.60
nM
Dasatinib TXK 2.10
nM
Dasatinib GAK 2.60
nM
Dasatinib KIT(D816V) 2.60
nM
Dasatinib KIT(V559D,V654A) 2.70
nM
Dasatinib DDR2 3.20
nM
Dasatinib MP2K5 3.30
nM