Dasatinib KINOMEscan - Dataset (ID:20196)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Dasatinib | EPHB2 | 0.39 | nM |
Dasatinib | EPHB1 | 0.45 | nM |
Dasatinib | PGFRA | 0.47 | nM |
Dasatinib | FGR | 0.50 | nM |
Dasatinib | KIT(L576P) | 0.57 | nM |
Dasatinib | LYN | 0.57 | nM |
Dasatinib | CSF1R | 0.58 | nM |
Dasatinib | PGFRB | 0.63 | nM |
Dasatinib | KIT(A829P) | 0.66 | nM |
Dasatinib | KIT(V559D) | 0.68 | nM |
Dasatinib | DDR1 | 0.69 | nM |
Dasatinib | FYN | 0.79 | nM |
Dasatinib | KIT | 0.81 | nM |
Dasatinib | EPHA2 | 0.85 | nM |
Dasatinib | CSK | 1.00 | nM |
Dasatinib | EPHA4 | 1.20 | nM |
Dasatinib | BMX | 1.40 | nM |
Dasatinib | BTK | 1.40 | nM |
Dasatinib | KIT(D816H) | 1.60 | nM |
Dasatinib | TXK | 2.10 | nM |
Dasatinib | GAK | 2.60 | nM |
Dasatinib | KIT(D816V) | 2.60 | nM |
Dasatinib | KIT(V559D,V654A) | 2.70 | nM |
Dasatinib | DDR2 | 3.20 | nM |
Dasatinib | MP2K5 | 3.30 | nM |