HKI-272 KINOMEscan-2 - Dataset (ID:20195)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Neratinib | TIE1 | 390.0 | nM |
| Neratinib | MERTK | 400.0 | nM |
| Neratinib | M3K2 | 450.0 | nM |
| Neratinib | HCK | 490.0 | nM |
| Neratinib | FER | 510.0 | nM |
| Neratinib | MP2K7 | 530.0 | nM |
| Neratinib | CSK | 550.0 | nM |
| Neratinib | FES | 590.0 | nM |
| Neratinib | CSF1R | 670.0 | nM |
| Neratinib | TNK2 | 680.0 | nM |
| Neratinib | M3K13 | 740.0 | nM |
| Neratinib | LYN | 820.0 | nM |
| Neratinib | KPCD1 | 820.0 | nM |
| Neratinib | CHK2 | 850.0 | nM |
| Neratinib | STK33 | 940.0 | nM |
| Neratinib | KPCD2 | 1100.0 | nM |
| Neratinib | DRAK2 | 1100.0 | nM |
| Neratinib | WEE2 | 1300.0 | nM |
| Neratinib | HIPK4 | 1500.0 | nM |
| Neratinib | MLTK | 1500.0 | nM |
| Neratinib | NUAK1 | 1500.0 | nM |
| Neratinib | MELK | 1600.0 | nM |
| Neratinib | FGR | 1900.0 | nM |
| Neratinib | FAK1 | 1900.0 | nM |
| Neratinib | JAK3(JH1domain-catalytic) | 2000.0 | nM |