HKI-272 KINOMEscan-2 - Dataset (ID:20195)
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| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Neratinib | MAP3K4 | 39.0 | nM |
| Neratinib | MST2 | 58.0 | nM |
| Neratinib | MP2K5 | 63.0 | nM |
| Neratinib | SLK | 66.0 | nM |
| Neratinib | PAK2 | 79.0 | nM |
| Neratinib | BLK | 85.0 | nM |
| Neratinib | M4K1 | 93.0 | nM |
| Neratinib | GCN2(Kin.Dom.2,S808G) | 96.0 | nM |
| Neratinib | LCK | 120.0 | nM |
| Neratinib | MAP3K3 | 130.0 | nM |
| Neratinib | SNARK | 140.0 | nM |
| Neratinib | TNIK | 140.0 | nM |
| Neratinib | BTK | 160.0 | nM |
| Neratinib | AXL | 190.0 | nM |
| Neratinib | PAK1 | 210.0 | nM |
| Neratinib | SIK1 | 220.0 | nM |
| Neratinib | MAP4K2 | 220.0 | nM |
| Neratinib | YES | 240.0 | nM |
| Neratinib | GAK | 250.0 | nM |
| Neratinib | NEK2 | 250.0 | nM |
| Neratinib | MST1 | 270.0 | nM |
| Neratinib | CSNK1E | 290.0 | nM |
| Neratinib | MAP4K4 | 330.0 | nM |
| Neratinib | DRAK1 | 340.0 | nM |
| Neratinib | M3K12 | 370.0 | nM |