HKI-272 KINOMEscan-2 - Dataset (ID:20195)

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Small Molecule Protein Kd Conc unit
Neratinib MAP3K4 39.0
nM
Neratinib MAP4K2 220.0
nM
Neratinib M4K3 7.7
nM
Neratinib MAP4K4 330.0
nM
Neratinib MAP4K5 0.7
nM
Neratinib MAPKAPK2
nM
Neratinib MAPKAPK5
nM
Neratinib MARK1
nM
Neratinib MARK2
nM
Neratinib MARK3
nM
Neratinib MARK4
nM
Neratinib MAST1 5500.0
nM
Neratinib MP2K1 14.0
nM
Neratinib MP2K2 26.0
nM
Neratinib MP2K3
nM
Neratinib MP2K4
nM
Neratinib MP2K5 63.0
nM
Neratinib MP2K6
nM
Neratinib MELK 1600.0
nM
Neratinib MERTK 400.0
nM
Neratinib MET 4000.0
nM
Neratinib MET(M1250T) 6700.0
nM
Neratinib MET(Y1235D) 4200.0
nM
Neratinib MINK 29.0
nM
Neratinib MP2K7 530.0
nM