GSK-461364A KINOMEscan - Dataset (ID:20194)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
GSK461364 | IKKB | nM | |
GSK461364 | IKKE | nM | |
GSK461364 | INSR | nM | |
GSK461364 | INSRR | nM | |
GSK461364 | IRAK1 | 6400.0 | nM |
GSK461364 | IRAK3 | 3500.0 | nM |
GSK461364 | IRAK4 | nM | |
GSK461364 | ITK | nM | |
GSK461364 | JAK1(JH1domain-catalytic) | nM | |
GSK461364 | JAK1(JH2domain-pseudokinase) | nM | |
GSK461364 | JAK2(JH1domain-catalytic) | nM | |
GSK461364 | JAK3(JH1domain-catalytic) | nM | |
GSK461364 | JNK1 | nM | |
GSK461364 | JNK3 | nM | |
GSK461364 | KC1G1 | nM | |
GSK461364 | KC1G2 | nM | |
GSK461364 | KCC2D | 620.0 | nM |
GSK461364 | KCC4 | nM | |
GSK461364 | KGP1 | nM | |
GSK461364 | KGP2 | nM | |
GSK461364 | KIT | nM | |
GSK461364 | KIT(A829P) | 7200.0 | nM |
GSK461364 | KIT(D816H) | nM | |
GSK461364 | KIT(D816V) | 1600.0 | nM |
GSK461364 | KIT(L576P) | nM |