Sorafenib KINOMEscan-2 - Dataset (ID:20192)
Proteins Studied
Download: Excel (XLSX), Comma-separated (CSV)
LINCS ID | Name | HMS LINCS ID | UniProt ID | Alternative Names | Provider | Mutation | Phosphlorylation State | Domain | Protein Description |
---|---|---|---|---|---|---|---|---|---|
200176 | FRK | 200176 | P42685 | Tyrosine-protein kinase FRK; Fyn-related kinase; FRK; GTK; PTK5; RAK | KINOMEscan | Wild Type; Partial length | |||
200175 | FLT4 | 200175 | P35916 | Fms-related tyrosine kinase 4; FLT4; FLT41; LMPH1A; PCL; VEGFR3 | KINOMEscan | Wild Type; Partial length | |||
200174 | FLT3(R834Q) | 200174 | P36888 | Fms-related tyrosine kinase 3; CD135; FLK2; FLK-2; FLT3; FLT-3; Ly72; STK1 | KINOMEscan | R834Q | Mutation (R834Q); Partial length | ||
200173 | FLT3(N841I) | 200173 | P36888 | Fms-related tyrosine kinase 3; CD135; FLK2; FLK-2; FLT3; FLT-3; Ly72; STK1 | KINOMEscan | N841I | Mutation (N841I); Partial length | ||
200172 | FLT3(K663Q) | 200172 | P36888 | Fms-related tyrosine kinase 3; CD135; FLK2; FLK-2; FLT3; FLT-3; Ly72; STK1 | KINOMEscan | K663Q | Mutation (K663Q); Partial length | ||
200171 | FLT3(ITD) | 200171 | P36888 | Fms-related tyrosine kinase 3; CD135; FLK2; FLK-2; FLT3; FLT-3; Ly72; STK1 | KINOMEscan | ITD | Mutation (ITD); Partial length | ||
200170 | FLT3(D835Y) | 200170 | P36888 | Fms-related tyrosine kinase 3; CD135; FLK2; FLK-2; FLT3; FLT-3; Ly72; STK1 | KINOMEscan | D835Y | Mutation (D835Y); Partial length | ||
200169 | FLT3(D835H) | 200169 | P36888 | Fms-related tyrosine kinase 3; CD135; FLK2; FLK-2; FLT3; FLT-3; Ly72; STK1 | KINOMEscan | D835H | Mutation (D835H); Partial length | ||
200168 | FLT3 | 200168 | P36888 | Fms-related tyrosine kinase 3; CD135; FLK2; FLK-2; FLT3; FLT-3; Ly72; STK1 | KINOMEscan | Wild Type; Partial length | |||
200167 | VGFR1 | 200167 | P17948 | Vascular endothelial growth factor receptor 1; fms-related tyrosine kinase 1; vascular permeability factor receptor; FLT; FLT1; VEGFR1 | KINOMEscan | Wild Type; Partial length | |||
200166 | FGR | 200166 | P09769 | Gardner-Rasheed feline sarcoma viral (v-fgr) oncogene homolog; c-fgr; c-src2; FGR; FLJ43153; MGC75096; p55c-fgr; p55-Fgr; p58c-fgr; SRC2 | KINOMEscan | Wild Type; Partial length | |||
200165 | FGFR4 | 200165 | P22455 | Fibroblast growth factor receptor 4; CD334; FGFR4; JTK2; MGC20292; TKF | KINOMEscan | Wild Type; Partial length | |||
200164 | FGFR3(G697C) | 200164 | P22607 | Fibroblast growth factor receptor 3; ACH; CD333; CEK2; FGFR3; HSFGFR3EX; JTK4 | KINOMEscan | G697C | Mutation (G697C); Partial length | ||
200163 | FGFR3 | 200163 | P22607 | Fibroblast growth factor receptor 3; ACH; CD333; CEK2; FGFR3; HSFGFR3EX; JTK4 | KINOMEscan | Wild Type; Partial length | |||
200162 | FGFR2 | 200162 | P21802 | Fibroblast growth factor receptor 2; BEK; BFR-1; CD332; CEK3; CFD1; ECT1; FGFR2; FLJ98662; JWS; KGFR; K-SAM; TK14; TK25 | KINOMEscan | Wild Type; Partial length | |||
200161 | FGFR1 | 200161 | P11362 | Fibroblast growth factor receptor 1; BFGFR; CD331; CEK; FGFBR; FGFR1; FLG; FLJ99988; FLT2; HBGFR; KAL2; N-SAM; OGD | KINOMEscan | Wild Type; Partial length | |||
200160 | FES | 200160 | P07332 | Feline sarcoma oncogene; FES; FPS | KINOMEscan | Wild Type; Partial length | |||
200159 | FER | 200159 | P16591 | Fer (fps/fes related) tyrosine kinase; FER; TYK3 | KINOMEscan | Wild Type; Partial length | |||
200158 | FAK1 | 200158 | Q05397 | PTK2 protein tyrosine kinase 2; FADK; FAK; FAK1; FRNK; pp125FAK; PTK2 | KINOMEscan | Wild Type; Partial length | |||
200157 | ERN1 | 200157 | O75460 | Endoplasmic reticulum to nucleus signaling 1; ERN1; FLJ30999; hIRE1p; IRE1; IRE1a; IRE1P; MGC163277; MGC163279 | KINOMEscan | Wild Type; Partial length | |||
200156 | ERK8 | 200156 | Q8TD08 | Mitogen-activated protein kinase 15; ERK7; ERK8; MAPK15 | KINOMEscan | Wild Type; Partial length | |||
200155 | ERK5 | 200155 | Q13164 | Mitogen-activated protein kinase 7; BMK1; ERK4; ERK5; MAPK7; PRKM7 | KINOMEscan | Wild Type; Partial length | |||
200154 | ERK4 | 200154 | P31152 | Mitogen-activated protein kinase 4; ERK3; Erk4; MAPK4; p63MAPK; PRKM4 | KINOMEscan | Wild Type; Partial length | |||
200153 | ERK3 | 200153 | Q16659 | Mitogen-activated protein kinase 6; DKFZp686F03189; ERK3; HsT17250; MAPK6; p97MAPK; PRKM6 | KINOMEscan | Wild Type; Partial length | |||
200152 | MK01 | 200152 | P28482 | Mitogen-activated protein kinase 1; ERK; ERK2; ERT1; MAPK1; MAPK2; p38; p40; p41; p41mapk; P42MAPK; PRKM1; PRKM2 | KINOMEscan | Wild Type; Full length |