CEP-701 KINOMEscan - Dataset (ID:20189)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Lestaurtinib | PHKG1 | 0.4 | nM |
Lestaurtinib | YSK4 | 0.5 | nM |
Lestaurtinib | FLT3(D835Y) | 0.6 | nM |
Lestaurtinib | FLT3(D835H) | 0.7 | nM |
Lestaurtinib | LATS2 | 1.0 | nM |
Lestaurtinib | SNARK | 1.0 | nM |
Lestaurtinib | FLT3(N841I) | 1.4 | nM |
Lestaurtinib | MKNK2 | 1.4 | nM |
Lestaurtinib | PLK4 | 1.5 | nM |
Lestaurtinib | FLT3(ITD) | 1.5 | nM |
Lestaurtinib | IRAK4 | 1.7 | nM |
Lestaurtinib | PHKG2 | 1.7 | nM |
Lestaurtinib | PKN2 | 1.8 | nM |
Lestaurtinib | JAK3(JH1domain-catalytic) | 2.3 | nM |
Lestaurtinib | MST2 | 2.4 | nM |
Lestaurtinib | LRRK2(G2019S) | 2.5 | nM |
Lestaurtinib | CHEK1 | 2.8 | nM |
Lestaurtinib | TAK1 | 2.9 | nM |
Lestaurtinib | CLK4 | 3.0 | nM |
Lestaurtinib | MST1 | 3.0 | nM |
Lestaurtinib | AAK1 | 3.1 | nM |
Lestaurtinib | DRAK1 | 3.4 | nM |
Lestaurtinib | PDPK1 | 3.4 | nM |
Lestaurtinib | MAP3K15 | 3.4 | nM |
Lestaurtinib | MLK1 | 3.5 | nM |