Vandetanib KINOMEscan - Dataset (ID:20186)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Vandetanib | RIPK2 | 4.6 | nM |
Vandetanib | EGFR(E746-A750del) | 4.8 | nM |
Vandetanib | EGFR(G719S) | 5.9 | nM |
Vandetanib | EGFR(L747-S752del, P753S) | 7.9 | nM |
Vandetanib | EGFR(L858R) | 8.7 | nM |
Vandetanib | EGFR(L747-T751del,Sins) | 8.9 | nM |
Vandetanib | ABL1(Y253F)-phosphorylated | 9.0 | nM |
Vandetanib | EGFR | 9.5 | nM |
Vandetanib | EGFR(G719C) | 9.6 | nM |
Vandetanib | ABL1(H396P)-nonphosphorylated | 9.8 | nM |
Vandetanib | DDR1 | 11.0 | nM |
Vandetanib | EGFR(L861Q) | 11.0 | nM |
Vandetanib | EGFR(S752-I759del) | 12.0 | nM |
Vandetanib | EGFR(L747-E749del, A750P) | 12.0 | nM |
Vandetanib | ABL1(E255K)-phosphorylated | 13.0 | nM |
Vandetanib | RET(M918T) | 14.0 | nM |
Vandetanib | ABL1(H396P)-phosphorylated | 14.0 | nM |
Vandetanib | ABL1(M351T)-phosphorylated | 15.0 | nM |
Vandetanib | ABL1(Q252H)-phosphorylated | 16.0 | nM |
Vandetanib | ABL1-phosphorylated | 16.0 | nM |
Vandetanib | LCK | 17.0 | nM |
Vandetanib | ABL1(Q252H)-nonphosphorylated | 18.0 | nM |
Vandetanib | ABL1(T315I)-phosphorylated | 20.0 | nM |
Vandetanib | ABL1(F317L)-phosphorylated | 33.0 | nM |
Vandetanib | RET | 34.0 | nM |