KW-2449 KINOMEscan - Dataset (ID:20185)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
KW2449 | IKKB | 430.0 | nM |
KW2449 | IKKE | 340.0 | nM |
KW2449 | INSR | 400.0 | nM |
KW2449 | INSRR | 420.0 | nM |
KW2449 | IRAK1 | 48.0 | nM |
KW2449 | IRAK3 | 240.0 | nM |
KW2449 | IRAK4 | 680.0 | nM |
KW2449 | ITK | 240.0 | nM |
KW2449 | JAK1(JH1domain-catalytic) | 1200.0 | nM |
KW2449 | JAK1(JH2domain-pseudokinase) | 190.0 | nM |
KW2449 | JAK2(JH1domain-catalytic) | 76.0 | nM |
KW2449 | JAK3(JH1domain-catalytic) | 39.0 | nM |
KW2449 | JNK1 | 580.0 | nM |
KW2449 | JNK3 | 51.0 | nM |
KW2449 | KC1G1 | 1200.0 | nM |
KW2449 | KC1G2 | 580.0 | nM |
KW2449 | KCC2D | nM | |
KW2449 | KCC4 | nM | |
KW2449 | KGP1 | 2500.0 | nM |
KW2449 | KGP2 | 800.0 | nM |
KW2449 | KIT | 53.0 | nM |
KW2449 | KIT(A829P) | 860.0 | nM |
KW2449 | KIT(D816H) | 240.0 | nM |
KW2449 | KIT(D816V) | 160.0 | nM |
KW2449 | KIT(L576P) | 21.0 | nM |