GSK-1363089 KINOMEscan - Dataset (ID:20176)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Foretinib | FLT3(D835Y) | 2.0 | nM |
Foretinib | KIT(V559D) | 2.1 | nM |
Foretinib | KIT(V559D,T670I) | 2.4 | nM |
Foretinib | EPHA7 | 2.5 | nM |
Foretinib | KIT | 2.5 | nM |
Foretinib | MP2K5 | 2.5 | nM |
Foretinib | FLT3(ITD) | 2.6 | nM |
Foretinib | KIT(L576P) | 2.7 | nM |
Foretinib | RET(V804M) | 2.8 | nM |
Foretinib | SLK | 3.0 | nM |
Foretinib | MST1R | 3.0 | nM |
Foretinib | TIE2 | 3.1 | nM |
Foretinib | KIT(A829P) | 3.2 | nM |
Foretinib | TRKC | 3.4 | nM |
Foretinib | PLK4 | 3.5 | nM |
Foretinib | EPHA2 | 3.6 | nM |
Foretinib | DDR2 | 3.6 | nM |
Foretinib | MKNK2 | 3.7 | nM |
Foretinib | CDK7 | 3.7 | nM |
Foretinib | FRK | 3.8 | nM |
Foretinib | VGFR1 | 3.8 | nM |
Foretinib | EPHB2 | 3.9 | nM |
Foretinib | ABL1(Q252H)-nonphosphorylated | 4.0 | nM |
Foretinib | MAP4K5 | 4.0 | nM |
Foretinib | TRKB | 4.1 | nM |