GSK-1363089 KINOMEscan - Dataset (ID:20176)

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Small Molecule Protein Kd Conc unit
Foretinib FLT3(D835Y) 2.0
nM
Foretinib KIT(V559D) 2.1
nM
Foretinib KIT(V559D,T670I) 2.4
nM
Foretinib EPHA7 2.5
nM
Foretinib KIT 2.5
nM
Foretinib MP2K5 2.5
nM
Foretinib FLT3(ITD) 2.6
nM
Foretinib KIT(L576P) 2.7
nM
Foretinib RET(V804M) 2.8
nM
Foretinib SLK 3.0
nM
Foretinib MST1R 3.0
nM
Foretinib TIE2 3.1
nM
Foretinib KIT(A829P) 3.2
nM
Foretinib TRKC 3.4
nM
Foretinib PLK4 3.5
nM
Foretinib EPHA2 3.6
nM
Foretinib DDR2 3.6
nM
Foretinib MKNK2 3.7
nM
Foretinib CDK7 3.7
nM
Foretinib FRK 3.8
nM
Foretinib VGFR1 3.8
nM
Foretinib EPHB2 3.9
nM
Foretinib ABL1(Q252H)-nonphosphorylated 4.0
nM
Foretinib MAP4K5 4.0
nM
Foretinib TRKB 4.1
nM