TG-101348 KINOMEscan - Dataset (ID:20174)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Fedratinib | CAMK1G | 3200.0 | nM |
Fedratinib | TESK1 | 3200.0 | nM |
Fedratinib | MLK1 | 3200.0 | nM |
Fedratinib | EGFR(L858R) | 3300.0 | nM |
Fedratinib | EGFR | 3400.0 | nM |
Fedratinib | NEK1 | 3400.0 | nM |
Fedratinib | MP2K3 | 3500.0 | nM |
Fedratinib | KIT(V559D,V654A) | 3500.0 | nM |
Fedratinib | ZAP70 | 3800.0 | nM |
Fedratinib | CHEK1 | 3800.0 | nM |
Fedratinib | KGP1 | 3800.0 | nM |
Fedratinib | PAK4 | 3800.0 | nM |
Fedratinib | EGFR(L747-T751del,Sins) | 3800.0 | nM |
Fedratinib | EPHB2 | 3900.0 | nM |
Fedratinib | EPHA6 | 3900.0 | nM |
Fedratinib | PIK3CA(H1047L) | 3900.0 | nM |
Fedratinib | EPHA4 | 4000.0 | nM |
Fedratinib | CAMKK2 | 4000.0 | nM |
Fedratinib | MAP3K4 | 4100.0 | nM |
Fedratinib | PI42C | 4100.0 | nM |
Fedratinib | ANKK1 | 4300.0 | nM |
Fedratinib | VGFR1 | 4300.0 | nM |
Fedratinib | AURKA | 4400.0 | nM |
Fedratinib | RPS6KA5(Kin.Dom.1-N-terminal) | 4400.0 | nM |
Fedratinib | MET(M1250T) | 4400.0 | nM |