PI-103 KINOMEscan - Dataset (ID:20167)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
PI103 | PIK3CA(C420R) | 1.3 | nM |
PI103 | PIK3CA(E542K) | 1.4 | nM |
PI103 | PIK3CA(E545K) | 1.5 | nM |
PI103 | PIK3CA | 1.5 | nM |
PI103 | PIK3CA(Q546K) | 1.5 | nM |
PI103 | PIK3CA(E545A) | 1.5 | nM |
PI103 | PIK3CB | 1.7 | nM |
PI103 | PIK3CA(I800L) | 2.9 | nM |
PI103 | PIK3CA(M1043I) | 3.0 | nM |
PI103 | PIK3CA(H1047L) | 3.2 | nM |
PI103 | PIK3CA(H1047Y) | 3.4 | nM |
PI103 | PIK3C2B | 10.0 | nM |
PI103 | MTOR | 12.0 | nM |
PI103 | PIK3CG | 16.0 | nM |
PI103 | PIK3CD | 17.0 | nM |
PI103 | PIK3C2G | 41.0 | nM |
PI103 | HIPK2 | 290.0 | nM |
PI103 | HIPK3 | 310.0 | nM |
PI103 | PI42C | 620.0 | nM |
PI103 | RIOK2 | 770.0 | nM |
PI103 | DAPK3 | 840.0 | nM |
PI103 | YSK4 | 930.0 | nM |
PI103 | MYLK | 1500.0 | nM |
PI103 | IKKA | 1700.0 | nM |
PI103 | MRCKA | 1800.0 | nM |