CI-1033 KINOMEscan-2 - Dataset (ID:20164)

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Small Molecule Protein Kd Conc unit
Canertinib LYN 810.00
nM
Canertinib MET(Y1235D) 830.00
nM
Canertinib RET(M918T) 840.00
nM
Canertinib ABL2 870.00
nM
Canertinib ABL1(F317I)-phosphorylated 1000.00
nM
Canertinib TYRO3 1000.00
nM
Canertinib LRRK2(G2019S) 1100.00
nM
Canertinib MK09 1100.00
nM
Canertinib SRC 1100.00
nM
Canertinib HIPK4 1100.00
nM
Canertinib FLT3(D835H) 1200.00
nM
Canertinib EPHA5 1200.00
nM
Canertinib MLTK 1200.00
nM
Canertinib IRAK4 1200.00
nM
Canertinib CIT 1300.00
nM
Canertinib ABL1(F317L)-nonphosphorylated 1500.00
nM
Canertinib EPHB1 1500.00
nM
Canertinib ADCK3 1500.00
nM
Canertinib TEC 1500.00
nM
Canertinib DYRK1A 1500.00
nM
Canertinib FLT3(K663Q) 1600.00
nM
Canertinib MP2K2 1600.00
nM
Canertinib BTK 1600.00
nM
Canertinib YES 1600.00
nM
Canertinib ERK3 1700.00
nM