CI-1033 KINOMEscan-2 - Dataset (ID:20164)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Canertinib | LYN | 810.00 | nM |
Canertinib | MET(Y1235D) | 830.00 | nM |
Canertinib | RET(M918T) | 840.00 | nM |
Canertinib | ABL2 | 870.00 | nM |
Canertinib | ABL1(F317I)-phosphorylated | 1000.00 | nM |
Canertinib | TYRO3 | 1000.00 | nM |
Canertinib | LRRK2(G2019S) | 1100.00 | nM |
Canertinib | MK09 | 1100.00 | nM |
Canertinib | SRC | 1100.00 | nM |
Canertinib | HIPK4 | 1100.00 | nM |
Canertinib | FLT3(D835H) | 1200.00 | nM |
Canertinib | EPHA5 | 1200.00 | nM |
Canertinib | MLTK | 1200.00 | nM |
Canertinib | IRAK4 | 1200.00 | nM |
Canertinib | CIT | 1300.00 | nM |
Canertinib | ABL1(F317L)-nonphosphorylated | 1500.00 | nM |
Canertinib | EPHB1 | 1500.00 | nM |
Canertinib | ADCK3 | 1500.00 | nM |
Canertinib | TEC | 1500.00 | nM |
Canertinib | DYRK1A | 1500.00 | nM |
Canertinib | FLT3(K663Q) | 1600.00 | nM |
Canertinib | MP2K2 | 1600.00 | nM |
Canertinib | BTK | 1600.00 | nM |
Canertinib | YES | 1600.00 | nM |
Canertinib | ERK3 | 1700.00 | nM |