CI-1033 KINOMEscan-2 - Dataset (ID:20164)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Canertinib | ABL1(Q252H)-nonphosphorylated | 91.00 | nM |
| Canertinib | GAK | 100.00 | nM |
| Canertinib | MP2K7 | 110.00 | nM |
| Canertinib | ABL1-nonphosphorylated | 210.00 | nM |
| Canertinib | ERBB3 | 210.00 | nM |
| Canertinib | MKNK1 | 260.00 | nM |
| Canertinib | EPHA6 | 270.00 | nM |
| Canertinib | RIPK2 | 300.00 | nM |
| Canertinib | LCK | 320.00 | nM |
| Canertinib | MAP4K2 | 330.00 | nM |
| Canertinib | DDR1 | 400.00 | nM |
| Canertinib | CSNK1E | 420.00 | nM |
| Canertinib | IRAK1 | 450.00 | nM |
| Canertinib | FLT3(R834Q) | 490.00 | nM |
| Canertinib | LRRK2 | 500.00 | nM |
| Canertinib | KIT(D816H) | 600.00 | nM |
| Canertinib | JAK3(JH1domain-catalytic) | 630.00 | nM |
| Canertinib | EPHB6 | 640.00 | nM |
| Canertinib | ABL1(T315I)-nonphosphorylated | 690.00 | nM |
| Canertinib | YSK4 | 700.00 | nM |
| Canertinib | TXK | 700.00 | nM |
| Canertinib | SIK3 | 700.00 | nM |
| Canertinib | KIT(A829P) | 700.00 | nM |
| Canertinib | FLT3(D835Y) | 730.00 | nM |
| Canertinib | TGFBR2 | 800.00 | nM |