CI-1033 KINOMEscan-2 - Dataset (ID:20164)

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Small Molecule Protein Kd Conc unit
Canertinib PGFRA 5200.00
nM
Canertinib LTK 5100.00
nM
Canertinib SIK2 4900.00
nM
Canertinib ULK3 4700.00
nM
Canertinib CSNK1D 4600.00
nM
Canertinib STK36 4500.00
nM
Canertinib RET 4200.00
nM
Canertinib HCK 4200.00
nM
Canertinib AURKB 4200.00
nM
Canertinib KIT(D816V) 3900.00
nM
Canertinib PTK6 3800.00
nM
Canertinib M3K2 3800.00
nM
Canertinib BIKE 3800.00
nM
Canertinib EPHA4 3600.00
nM
Canertinib ADCK4 3400.00
nM
Canertinib FRK 3400.00
nM
Canertinib TAK1 3300.00
nM
Canertinib TESK1 3200.00
nM
Canertinib ABL1(F317I)-nonphosphorylated 3200.00
nM
Canertinib FLT3(ITD) 3000.00
nM
Canertinib IRAK3 3000.00
nM
Canertinib STK35 2900.00
nM
Canertinib FGR 2800.00
nM
Canertinib AURKC 2800.00
nM
Canertinib EPHB2 2700.00
nM