CI-1033 KINOMEscan-2 - Dataset (ID:20164)

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Small Molecule Protein Kd Conc unit
Canertinib KIT 7800.00
nM
Canertinib KIT(A829P) 700.00
nM
Canertinib KIT(D816H) 600.00
nM
Canertinib KIT(D816V) 3900.00
nM
Canertinib KIT(L576P) 5700.00
nM
Canertinib KIT(V559D) 7900.00
nM
Canertinib KIT(V559D,T670I) 1900.00
nM
Canertinib KIT(V559D,V654A) 7900.00
nM
Canertinib LATS1
nM
Canertinib LATS2
nM
Canertinib LCK 320.00
nM
Canertinib LIMK1
nM
Canertinib LIMK2
nM
Canertinib LKB1
nM
Canertinib LOK 1900.00
nM
Canertinib LRRK2 500.00
nM
Canertinib LRRK2(G2019S) 1100.00
nM
Canertinib LTK 5100.00
nM
Canertinib LYN 810.00
nM
Canertinib M3K13
nM
Canertinib MAK
nM
Canertinib MAP3K1
nM
Canertinib MAP3K15
nM
Canertinib M3K2 3800.00
nM
Canertinib MAP3K3 2300.00
nM