CI-1033 KINOMEscan-2 - Dataset (ID:20164)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Canertinib | KIT | 7800.00 | nM |
Canertinib | KIT(A829P) | 700.00 | nM |
Canertinib | KIT(D816H) | 600.00 | nM |
Canertinib | KIT(D816V) | 3900.00 | nM |
Canertinib | KIT(L576P) | 5700.00 | nM |
Canertinib | KIT(V559D) | 7900.00 | nM |
Canertinib | KIT(V559D,T670I) | 1900.00 | nM |
Canertinib | KIT(V559D,V654A) | 7900.00 | nM |
Canertinib | LATS1 | nM | |
Canertinib | LATS2 | nM | |
Canertinib | LCK | 320.00 | nM |
Canertinib | LIMK1 | nM | |
Canertinib | LIMK2 | nM | |
Canertinib | LKB1 | nM | |
Canertinib | LOK | 1900.00 | nM |
Canertinib | LRRK2 | 500.00 | nM |
Canertinib | LRRK2(G2019S) | 1100.00 | nM |
Canertinib | LTK | 5100.00 | nM |
Canertinib | LYN | 810.00 | nM |
Canertinib | M3K13 | nM | |
Canertinib | MAK | nM | |
Canertinib | MAP3K1 | nM | |
Canertinib | MAP3K15 | nM | |
Canertinib | M3K2 | 3800.00 | nM |
Canertinib | MAP3K3 | 2300.00 | nM |