Nilotinib KINOMEscan - Dataset (ID:20162)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Nilotinib | DDR1 | 1.1 | nM |
Nilotinib | ABL1(H396P)-nonphosphorylated | 4.9 | nM |
Nilotinib | ABL1(Q252H)-nonphosphorylated | 10.0 | nM |
Nilotinib | ABL1-nonphosphorylated | 10.0 | nM |
Nilotinib | MLTK | 11.0 | nM |
Nilotinib | ABL1(F317L)-nonphosphorylated | 12.0 | nM |
Nilotinib | ABL1(Y253F)-phosphorylated | 13.0 | nM |
Nilotinib | ABL1-phosphorylated | 13.0 | nM |
Nilotinib | ABL1(F317L)-phosphorylated | 14.0 | nM |
Nilotinib | ABL1(M351T)-phosphorylated | 15.0 | nM |
Nilotinib | ABL1(F317I)-nonphosphorylated | 18.0 | nM |
Nilotinib | ABL1(Q252H)-phosphorylated | 21.0 | nM |
Nilotinib | ABL1(H396P)-phosphorylated | 21.0 | nM |
Nilotinib | KIT(L576P) | 22.0 | nM |
Nilotinib | ABL2 | 26.0 | nM |
Nilotinib | KIT | 29.0 | nM |
Nilotinib | DDR2 | 33.0 | nM |
Nilotinib | MK11 | 36.0 | nM |
Nilotinib | ABL1(E255K)-phosphorylated | 36.0 | nM |
Nilotinib | EPHA8 | 37.0 | nM |
Nilotinib | CSF1R | 45.0 | nM |
Nilotinib | KIT(V559D) | 46.0 | nM |
Nilotinib | KIT(A829P) | 46.0 | nM |
Nilotinib | LCK | 47.0 | nM |
Nilotinib | ABL1(F317I)-phosphorylated | 56.0 | nM |