LY-317615 KINOMEscan - Dataset (ID:20159)
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| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Enzastaurin | GSK3B | 8.3 | nM |
| Enzastaurin | KPCE | 8.9 | nM |
| Enzastaurin | KPCD | 25.0 | nM |
| Enzastaurin | RSK4(Kin.Dom.1-N-terminal) | 25.0 | nM |
| Enzastaurin | KPCT | 36.0 | nM |
| Enzastaurin | FLT3(D835Y) | 40.0 | nM |
| Enzastaurin | KPCL | 46.0 | nM |
| Enzastaurin | FLT3(D835H) | 49.0 | nM |
| Enzastaurin | FLT3(ITD) | 72.0 | nM |
| Enzastaurin | ERK8 | 76.0 | nM |
| Enzastaurin | RSK2(Kin.Dom.1-N-terminal) | 87.0 | nM |
| Enzastaurin | DYRK1A | 160.0 | nM |
| Enzastaurin | KGP2 | 170.0 | nM |
| Enzastaurin | PIM1 | 200.0 | nM |
| Enzastaurin | RSK3(Kin.Dom.1-N-terminal) | 220.0 | nM |
| Enzastaurin | MYLK4 | 230.0 | nM |
| Enzastaurin | FLT3(N841I) | 250.0 | nM |
| Enzastaurin | FLT3 | 330.0 | nM |
| Enzastaurin | PKAC-alpha | 330.0 | nM |
| Enzastaurin | RPS6KA5(Kin.Dom.1-N-terminal) | 370.0 | nM |
| Enzastaurin | FLT3(K663Q) | 420.0 | nM |
| Enzastaurin | CLK2 | 430.0 | nM |
| Enzastaurin | TLK1 | 510.0 | nM |
| Enzastaurin | CLK1 | 510.0 | nM |
| Enzastaurin | PKAC-beta | 590.0 | nM |