AZD-6244 KINOMEscan - Dataset (ID:20156)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Selumetinib | MP2K1 | 99.0 | nM |
Selumetinib | MP2K2 | 530.0 | nM |
Selumetinib | EGFR(T790M) | 2200.0 | nM |
Selumetinib | EGFR(L747-E749del, A750P) | 3000.0 | nM |
Selumetinib | EGFR(G719C) | 4200.0 | nM |
Selumetinib | EGFR(S752-I759del) | 5000.0 | nM |
Selumetinib | EGFR(G719S) | 5200.0 | nM |
Selumetinib | EGFR(L747-S752del, P753S) | 5300.0 | nM |
Selumetinib | EGFR(L747-T751del,Sins) | 5500.0 | nM |
Selumetinib | EGFR(E746-A750del) | 5700.0 | nM |
Selumetinib | EGFR | 7000.0 | nM |
Selumetinib | EGFR(L858R) | 8000.0 | nM |
Selumetinib | EGFR(L861Q) | 8900.0 | nM |
Selumetinib | ABL1-nonphosphorylated | nM | |
Selumetinib | ABL1(Y253F)-phosphorylated | nM | |
Selumetinib | ABL1(H396P)-nonphosphorylated | nM | |
Selumetinib | ABL1(T315I)-phosphorylated | nM | |
Selumetinib | ABL1(T315I)-nonphosphorylated | nM | |
Selumetinib | ABL1(F317L)-phosphorylated | nM | |
Selumetinib | ABL1(F317I)-nonphosphorylated | nM | |
Selumetinib | ADCK3 | nM | |
Selumetinib | ACVRL1 | nM | |
Selumetinib | ADCK4 | nM | |
Selumetinib | ABL1(Q252H)-phosphorylated | nM | |
Selumetinib | ACVR2B | nM |