AC220 KINOMEscan - Dataset (ID:20147)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| AC220 | FLT3 | 1.3 | nM |
| AC220 | FLT3(K663Q) | 2.2 | nM |
| AC220 | RET(M918T) | 3.0 | nM |
| AC220 | KIT(A829P) | 3.6 | nM |
| AC220 | FLT3(D835H) | 3.7 | nM |
| AC220 | FLT3(N841I) | 4.1 | nM |
| AC220 | KIT | 4.8 | nM |
| AC220 | KIT(V559D) | 5.0 | nM |
| AC220 | FLT3(R834Q) | 5.1 | nM |
| AC220 | KIT(V559D,T670I) | 6.0 | nM |
| AC220 | KIT(L576P) | 6.3 | nM |
| AC220 | FLT3(D835Y) | 7.1 | nM |
| AC220 | PGFRB | 7.7 | nM |
| AC220 | RET | 8.0 | nM |
| AC220 | FLT3(ITD) | 8.8 | nM |
| AC220 | RET(V804M) | 9.1 | nM |
| AC220 | CSF1R | 10.0 | nM |
| AC220 | PGFRA | 11.0 | nM |
| AC220 | RET(V804L) | 13.0 | nM |
| AC220 | KIT(V559D,V654A) | 36.0 | nM |
| AC220 | VGFR1 | 41.0 | nM |
| AC220 | FLT4 | 41.0 | nM |
| AC220 | DDR1 | 81.0 | nM |
| AC220 | VGFR2 | 87.0 | nM |
| AC220 | KIT(D816V) | 150.0 | nM |