Breast cell line dose response to target inhibition measured by high throughput microscopy - Dataset (ID:20136)
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Small Molecule | Cell Line | Drug Concentration | Conc Units | Timepoint | Timepoint Units | Measured pERK (Alexa 488) | Measured p-Rb (Alexa 568) | Alexa Fluor 647 | Measured p-Akt/p-4EBP1/p-S6 (Alexa 647) | Image |
---|---|---|---|---|---|---|---|---|---|---|
Torkinib | MCF 10A | 0.1 | nM | 24 | hr | 422.39 | 160.17 | p-S6 | 363.48 | |
Torkinib | HCC1954 | 0.1 | nM | 6 | hr | 184.48 | 44.56 | p-S6 | 110.17 | |
Torkinib | HCC1954 | 0.1 | nM | 24 | hr | 274.70 | 113.00 | p-S6 | 380.78 | |
Torkinib | HCC1954 | 0.1 | nM | 24 | hr | 291.18 | 108.05 | p-S6 | 406.86 | |
Torkinib | MCF 10A | 0.1 | nM | 6 | hr | 500.23 | 174.95 | p-S6 | 699.38 | |
Torkinib | AU565 | 0.1 | nM | 24 | hr | 484.31 | 116.72 | p-Akt | 84.98 | |
Torkinib | HCC1954 | 0.1 | nM | 6 | hr | 195.86 | 37.51 | p-Akt | 23.03 | |
Torkinib | MCF 10A | 0.1 | nM | 6 | hr | 458.56 | 155.16 | p-Akt | 49.17 | |
Torkinib | MCF 10A | 0.1 | nM | 24 | hr | 342.29 | 124.00 | p-Akt | 50.29 | |
Torkinib | AU565 | 0.1 | nM | 6 | hr | 249.91 | 55.55 | p-Akt | 24.44 | |
Torkinib | AU565 | 0.1 | nM | 24 | hr | 513.30 | 118.22 | p-Akt | 83.59 | |
Torkinib | HCC1954 | 0.1 | nM | 24 | hr | 300.36 | 112.32 | p-Akt | 67.70 | |
Torkinib | MCF 10A | 0.1 | nM | 6 | hr | 483.02 | 168.09 | p-Akt | 48.88 | |
Torkinib | AU565 | 0.1 | nM | 6 | hr | 346.86 | 73.14 | p-4EBP1 | 98.91 | |
Torkinib | AU565 | 0.1 | nM | 24 | hr | 484.96 | 127.02 | p-4EBP1 | 215.15 | |
Torkinib | HCC1954 | 0.1 | nM | 24 | hr | 268.67 | 120.63 | p-4EBP1 | 124.48 | |
Torkinib | MCF 10A | 0.1 | nM | 6 | hr | 452.64 | 159.11 | p-4EBP1 | 351.84 | |
Torkinib | T47D | 0.1 | nM | 24 | hr | 157.07 | 112.77 | p-4EBP1 | 421.70 | |
Torkinib | AU565 | 0.1 | nM | 6 | hr | 226.90 | 50.34 | p-4EBP1 | 59.83 | |
Torkinib | HCC1954 | 0.1 | nM | 6 | hr | 179.96 | 38.18 | p-4EBP1 | 49.70 | |
Torkinib | HCC1954 | 0.1 | nM | 24 | hr | 294.96 | 117.90 | p-4EBP1 | 132.58 | |
Torkinib | AU565 | 0.1 | nM | 6 | hr | 230.65 | 52.24 | p-Akt | 23.88 | |
Torkinib | AU565 | 0.1 | nM | 6 | hr | 259.18 | 62.54 | p-S6 | 155.57 | |
Torkinib | MCF 10A | 0.422 | nM | 6 | hr | 430.95 | 160.56 | p-S6 | 549.49 | |
Torkinib | HCC1954 | 0.422 | nM | 24 | hr | 288.79 | 112.90 | p-S6 | 376.36 |