Breast cell line dose response to target inhibition measured by high throughput microscopy - Dataset (ID:20136)
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Small Molecule | Cell Line | Drug Concentration | Conc Units | Timepoint | Timepoint Units | Measured pERK (Alexa 488) | Measured p-Rb (Alexa 568) | Alexa Fluor 647 | Measured p-Akt/p-4EBP1/p-S6 (Alexa 647) | Image |
---|---|---|---|---|---|---|---|---|---|---|
GSK1059615 | AU565 | 0 (control) | 24 | hr | 447.87 | 123.71 | p-4EBP1 | 188.29 | ||
GSK1059615 | AU565 | 0 (control) | 6 | hr | 234.34 | 56.31 | p-4EBP1 | 61.94 | ||
Torkinib | AU565 | 0 (control) | 24 | hr | 520.08 | 134.68 | p-4EBP1 | 226.94 | ||
Torkinib | AU565 | 0 (control) | 6 | hr | 294.05 | 67.35 | p-4EBP1 | 84.02 | ||
Gefitinib | AU565 | 0 (control) | 24 | hr | 597.19 | 141.39 | p-4EBP1 | 180.42 | ||
Gefitinib | AU565 | 0 (control) | 6 | hr | 226.23 | 50.86 | p-4EBP1 | 51.79 | ||
Dactolisib | T47D | 0 (control) | 24 | hr | 165.27 | 86.01 | p-Akt | 60.10 | ||
Dactolisib | T47D | 0 (control) | 6 | hr | 99.23 | 26.75 | p-Akt | 14.05 | ||
Triciribine | T47D | 0 (control) | 24 | hr | 186.87 | 92.32 | p-Akt | 71.34 | ||
Triciribine | T47D | 0 (control) | 6 | hr | 109.11 | 47.87 | p-Akt | 21.01 | ||
MK2206 | T47D | 0 (control) | 24 | hr | 176.28 | 99.14 | p-Akt | 70.51 | ||
MK2206 | T47D | 0 (control) | 6 | hr | 102.66 | 35.62 | p-Akt | 15.31 | ||
GSK1059615 | T47D | 0 (control) | 24 | hr | 168.24 | 91.00 | p-Akt | 67.96 | ||
GSK1059615 | T47D | 0 (control) | 6 | hr | 168.92 | 88.95 | p-Akt | 95.10 | ||
Torkinib | T47D | 0 (control) | 24 | hr | 176.46 | 94.89 | p-Akt | 74.20 | ||
Torkinib | T47D | 0 (control) | 6 | hr | 192.56 | 91.57 | p-Akt | 104.03 | ||
Gefitinib | T47D | 0 (control) | 24 | hr | 177.88 | 116.19 | p-Akt | 85.23 | ||
Gefitinib | T47D | 0 (control) | 6 | hr | 176.65 | 97.90 | p-Akt | 103.18 | ||
Dactolisib | MCF 10A | 0 (control) | 24 | hr | 351.94 | 125.18 | p-Akt | 50.36 | ||
Dactolisib | MCF 10A | 0 (control) | 6 | hr | 436.72 | 165.98 | p-Akt | 55.27 | ||
Triciribine | MCF 10A | 0 (control) | 24 | hr | 333.49 | 112.55 | p-Akt | 47.91 | ||
Triciribine | MCF 10A | 0 (control) | 6 | hr | 477.54 | 163.37 | p-Akt | 60.15 | ||
MK2206 | MCF 10A | 0 (control) | 24 | hr | 334.53 | 120.26 | p-Akt | 52.16 | ||
MK2206 | MCF 10A | 0 (control) | 6 | hr | 475.25 | 162.73 | p-Akt | 59.87 | ||
GSK1059615 | MCF 10A | 0 (control) | 24 | hr | 372.12 | 121.72 | p-Akt | 53.36 |