AZD 5438 KINOMEscan - Dataset (ID:20135)

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Small Molecule Protein % Control Assay compound conc Conc unit
AZD 5438 ABL1(F317L)-phosphorylated 55.0 10
uM
AZD 5438 ABL1(F317L)-nonphosphorylated 96.0 10
uM
AZD 5438 ABL1(F317I)-phosphorylated 78.0 10
uM
AZD 5438 ABL1(F317I)-nonphosphorylated 100.0 10
uM
AZD 5438 ABL1(E255K)-phosphorylated 6.3 10
uM
AZD 5438 AAK1 3.8 10
uM