Metrics other than potency reveal systematic variation in responses to cancer drugs - Dataset (ID:20120)
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Small Molecule | Cell Line | log10[max. dose (M)] | R^2 (goodness of fit) | log10[EC50 (M)] | log10[IC50 (M)] | log10[GI50 (M)] | HillSlope | E_inf | E_max | AUC |
---|---|---|---|---|---|---|---|---|---|---|
Tozasertib | HCC1569 | -4.0000 | 0.9023 | -5.0220 | -5.0220 | -5.7245 | 0.5522 | 0.0000 | 0.2143 | 6.7476 |
GSK461364 | HCC1569 | -4.4776 | 0.7965 | -5.0714 | -5.0714 | -5.7745 | 0.3696 | 0.0000 | 0.3763 | 6.5207 |
Tozasertib | HCC1395 | -4.0000 | 0.9267 | -4.9570 | -4.9570 | -5.7943 | 0.9915 | 0.0000 | 0.1011 | 6.6654 |
GSK461364 | T47D | -4.4776 | 0.7866 | -4.9834 | -4.9834 | -6.1129 | 1.8790 | 0.0000 | 0.1008 | 7.2108 |
GSK461364 | UACC-812 | -4.4776 | 0.8943 | -4.8642 | -4.8641 | -5.0359 | 3.7120 | 0.0000 | 0.0354 | 8.8806 |
Tozasertib | MDA-MB-134-VI | -4.0000 | 0.9695 | -4.7252 | -4.7252 | -5.7263 | 0.4520 | 0.0000 | 0.3198 | 7.0698 |
GSK461364 | LY2 | -4.4776 | 0.7525 | -5.3501 | -5.3501 | -5.9259 | 0.3841 | 0.0000 | 0.3161 | 6.7154 |
GSK461364 | 184B5 | -4.4776 | 0.7303 | -5.5881 | -5.5882 | -6.3658 | 0.4307 | 0.0000 | 0.2496 | 6.7499 |
Tozasertib | BT-474 | -4.0000 | 0.8143 | -4.4178 | -4.4177 | -5.1819 | 1.5550 | 0.0000 | 0.1831 | 7.9621 |
Tozasertib | MDA-MB-436 | -4.0000 | 0.8816 | -5.3890 | -5.3894 | -6.0657 | 0.4927 | 0.0000 | 0.1713 | 6.4739 |
GSK461364 | MCF 10F | -4.4776 | 0.8285 | -6.0156 | -6.0160 | -7.2051 | 0.4255 | 0.0000 | 0.2392 | 6.1498 |
Tozasertib | 184B5 | -4.0000 | 0.9641 | -5.3720 | -5.3719 | -5.7560 | 0.7204 | 0.0000 | 0.0932 | 6.4426 |
Tozasertib | MDA-MB-361 | -4.0000 | 0.9415 | -4.5904 | -4.5905 | -5.2826 | 2.2145 | 0.0000 | 0.0505 | 7.4753 |
Tozasertib | UACC-812 | -4.0000 | 0.8195 | -4.5034 | -4.5034 | -4.9544 | 1.8730 | 0.0000 | 0.1024 | 7.1924 |
GSK461364 | SUM185PE | -4.4776 | 0.8273 | -5.1574 | -5.1573 | -5.8411 | 1.7260 | 0.0000 | 0.0879 | 7.3788 |
Tozasertib | HCC70 | -4.0000 | 0.7843 | -5.2470 | -5.2466 | NaN | 0.3821 | 0.0000 | 0.2503 | 6.3077 |
Tozasertib | BT-20 | -4.0000 | 0.8366 | -4.6124 | -4.6124 | -5.5324 | 0.4999 | 0.0000 | 0.3307 | 7.0328 |
Tozasertib | MDA-MB-157 | -4.0000 | 0.9065 | -5.0270 | -5.0273 | -5.4475 | 0.8482 | 0.0000 | 0.1185 | 6.9191 |
GSK461364 | 184A1 | -4.4776 | 0.9640 | -4.8844 | -4.8844 | -5.2355 | 2.3020 | 0.0000 | 0.1037 | 7.8611 |
GSK461364 | MCF12A | -4.4776 | 0.7888 | -5.5836 | -5.5839 | -5.8310 | 0.4970 | 0.0000 | 0.2199 | 6.8984 |
Tozasertib | MDA-MB-231 | -4.0000 | 0.9221 | -4.8628 | -4.8630 | -4.9264 | 1.1070 | 0.0000 | 0.0998 | 7.3371 |
GSK461364 | BT-474 | -4.4776 | 0.7677 | -4.9305 | -4.9304 | -5.0842 | 3.9990 | 0.0000 | 0.0152 | 7.4055 |
GSK461364 | 600MPE | -4.4776 | 0.8618 | -4.8362 | -4.8362 | -4.8631 | 4.0000 | 0.0000 | 0.0355 | 7.9370 |
Imatinib | MDA-MB-134-VI | -3.2480 | 0.9236 | -4.2770 | -4.2771 | -4.5481 | 1.6620 | 0.0000 | 0.0191 | 6.5153 |
Imatinib | Hs 578T | -3.2480 | 0.7789 | -4.2235 | -4.2235 | -4.2478 | 3.9950 | 0.0000 | 0.0001 | 8.6178 |