NPK76-II-72-1 KiNativ -- single dose experiment - Dataset (ID:20106)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
NPK76-II-72-1 PC-3 IKKE,TBK1
DIkPGNIMR
Lys2
12.4
10
uM
NPK76-II-72-1 HeLa IKKE,TBK1
DIkPGNIMR
Lys2
-18.4
10
uM
NPK76-II-72-1 PC-3 LKB1
DIkPGNLLLTTGGTLK
Lys2
-14.1
10
uM
NPK76-II-72-1 HeLa LKB1
DIkPGNLLLTTGGTLK
Lys2
-8.7
10
uM
NPK76-II-72-1 PC-3 GSK3B
DIkPQNLLLDPDTAVLK
Lys2
-7.0
10
uM
NPK76-II-72-1 HeLa GSK3A
DIkPQNLLVDPDTAVLK
Lys2
-3.8
10
uM
NPK76-II-72-1 PC-3 MAP2K4
DIkPSNILLDR
Lys2
-11.5
10
uM
NPK76-II-72-1 PC-3 IRAK4
DIkSANILLDEAFTAK
Lys2
-8.9
10
uM
NPK76-II-72-1 HeLa IRAK4
DIkSANILLDEAFTAK
Lys2
-7.3
10
uM
NPK76-II-72-1 HeLa NEK1
DIkSQNIFLTK
Lys2
-0.3
10
uM
NPK76-II-72-1 PC-3 NEK9
DIkTLNIFLTK
Lys2
-7.8
10
uM
NPK76-II-72-1 HeLa NEK9
DIkTLNIFLTK
Lys2
-6.5
10
uM
NPK76-II-72-1 HeLa HPK1
DKVSGDLVALkMVK
Lys1
-23.2
10
uM
NPK76-II-72-1 PC-3 MARK2,MARK3
DLkAENLLLDADMNIK
Lys2
1.4
10
uM
NPK76-II-72-1 HeLa MARK2,MARK3
DLkAENLLLDADMNIK
Lys2
-44.8
10
uM
NPK76-II-72-1 HeLa SLK
DLkAGNILFTLDGDIK
Lys2
46.4
10
uM
NPK76-II-72-1 PC-3 SLK
DLkAGNILFTLDGDIK
Lys2
12.8
10
uM
NPK76-II-72-1 HeLa LOK
DLkAGNVLMTLEGDIR
Lys2
7.9
10
uM
NPK76-II-72-1 PC-3 LOK
DLkAGNVLMTLEGDIR
Lys2
-0.2
10
uM
NPK76-II-72-1 HeLa Wnk1,Wnk2,Wnk3
DLkCDNIFITGPTGSVK
Lys2
-9.3
10
uM
NPK76-II-72-1 PC-3 WNK4
DLkCDNVFITGPTGSVK
Lys2
3.0
10
uM
NPK76-II-72-1 HeLa BARK1
DLkPANILLDEHGHVR
Lys2
9.7
10
uM
NPK76-II-72-1 PC-3 CDK11,CDK8
DLkPANILVMGEGPER
Lys2
-14.6
10
uM
NPK76-II-72-1 HeLa MAST3
DLkPDNLLITSLGHIK
Lys2
5.7
10
uM
NPK76-II-72-1 PC-3 MAST3
DLkPDNLLITSLGHIK
Lys2
-7.8
10
uM