NPK76-II-72-1 KiNativ -- single dose experiment - Dataset (ID:20106)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
NPK76-II-72-1 | PC-3 | IKKE,TBK1 | DIkPGNIMR | Lys2 | 12.4 | 10 | uM |
NPK76-II-72-1 | HeLa | IKKE,TBK1 | DIkPGNIMR | Lys2 | -18.4 | 10 | uM |
NPK76-II-72-1 | PC-3 | LKB1 | DIkPGNLLLTTGGTLK | Lys2 | -14.1 | 10 | uM |
NPK76-II-72-1 | HeLa | LKB1 | DIkPGNLLLTTGGTLK | Lys2 | -8.7 | 10 | uM |
NPK76-II-72-1 | PC-3 | GSK3B | DIkPQNLLLDPDTAVLK | Lys2 | -7.0 | 10 | uM |
NPK76-II-72-1 | HeLa | GSK3A | DIkPQNLLVDPDTAVLK | Lys2 | -3.8 | 10 | uM |
NPK76-II-72-1 | PC-3 | MAP2K4 | DIkPSNILLDR | Lys2 | -11.5 | 10 | uM |
NPK76-II-72-1 | PC-3 | IRAK4 | DIkSANILLDEAFTAK | Lys2 | -8.9 | 10 | uM |
NPK76-II-72-1 | HeLa | IRAK4 | DIkSANILLDEAFTAK | Lys2 | -7.3 | 10 | uM |
NPK76-II-72-1 | HeLa | NEK1 | DIkSQNIFLTK | Lys2 | -0.3 | 10 | uM |
NPK76-II-72-1 | PC-3 | NEK9 | DIkTLNIFLTK | Lys2 | -7.8 | 10 | uM |
NPK76-II-72-1 | HeLa | NEK9 | DIkTLNIFLTK | Lys2 | -6.5 | 10 | uM |
NPK76-II-72-1 | HeLa | HPK1 | DKVSGDLVALkMVK | Lys1 | -23.2 | 10 | uM |
NPK76-II-72-1 | PC-3 | MARK2,MARK3 | DLkAENLLLDADMNIK | Lys2 | 1.4 | 10 | uM |
NPK76-II-72-1 | HeLa | MARK2,MARK3 | DLkAENLLLDADMNIK | Lys2 | -44.8 | 10 | uM |
NPK76-II-72-1 | HeLa | SLK | DLkAGNILFTLDGDIK | Lys2 | 46.4 | 10 | uM |
NPK76-II-72-1 | PC-3 | SLK | DLkAGNILFTLDGDIK | Lys2 | 12.8 | 10 | uM |
NPK76-II-72-1 | HeLa | LOK | DLkAGNVLMTLEGDIR | Lys2 | 7.9 | 10 | uM |
NPK76-II-72-1 | PC-3 | LOK | DLkAGNVLMTLEGDIR | Lys2 | -0.2 | 10 | uM |
NPK76-II-72-1 | HeLa | Wnk1,Wnk2,Wnk3 | DLkCDNIFITGPTGSVK | Lys2 | -9.3 | 10 | uM |
NPK76-II-72-1 | PC-3 | WNK4 | DLkCDNVFITGPTGSVK | Lys2 | 3.0 | 10 | uM |
NPK76-II-72-1 | HeLa | BARK1 | DLkPANILLDEHGHVR | Lys2 | 9.7 | 10 | uM |
NPK76-II-72-1 | PC-3 | CDK11,CDK8 | DLkPANILVMGEGPER | Lys2 | -14.6 | 10 | uM |
NPK76-II-72-1 | HeLa | MAST3 | DLkPDNLLITSLGHIK | Lys2 | 5.7 | 10 | uM |
NPK76-II-72-1 | PC-3 | MAST3 | DLkPDNLLITSLGHIK | Lys2 | -7.8 | 10 | uM |