NPK76-II-72-1 KiNativ -- single dose experiment - Dataset (ID:20106)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
NPK76-II-72-1 PC-3 SLK
ETSVLAAAkVIDTK
Lys1
68.4
10
uM
NPK76-II-72-1 HeLa SLK
DLkAGNILFTLDGDIK
Lys2
46.4
10
uM
NPK76-II-72-1 PC-3 SLK
DLkAGNILFTLDGDIK
Lys2
12.8
10
uM
NPK76-II-72-1 HeLa SMG1
DTVTIHSVGGTITILPTkTKPK
ATP
-7.2
10
uM
NPK76-II-72-1 PC-3 SRPK1
IIHTDIkPENILLSVNEQYIR
Lys2
14.4
10
uM
NPK76-II-72-1 HeLa STLK5
YSVkVLPWLSPEVLQQNLQGYDAK
Activation Loop
69.5
10
uM
NPK76-II-72-1 HeLa SYK
ISDFGLSkALR
Activation Loop
-12.9
10
uM
NPK76-II-72-1 HeLa TAO1,TAOK3
DIkAGNILLTEPGQVK
Lys2
-21.1
10
uM
NPK76-II-72-1 PC-3 TAO1,TAOK3
DIkAGNILLTEPGQVK
Lys2
-2.8
10
uM
NPK76-II-72-1 PC-3 TAOK2
DVkAGNILLSEPGLVK
Lys2
1.7
10
uM
NPK76-II-72-1 HeLa TBK1
TGDLFAIkVFNNISFLRPVDVQMR
Lys1
50.3
10
uM
NPK76-II-72-1 PC-3 TLK1
YAAVkIHQLNK
Lys1
-9.5
10
uM
NPK76-II-72-1 HeLa TLK1
YLNEIKPPIIHYDLkPGNILLVDGTACGEIK
Lys2
12.6
10
uM
NPK76-II-72-1 PC-3 TLK1
YLNEIKPPIIHYDLkPGNILLVDGTACGEIK
Lys2
-19.2
10
uM
NPK76-II-72-1 PC-3 TLK2
YVAVkIHQLNK
Lys1
-25.5
10
uM
NPK76-II-72-1 HeLa ULK1
DLkPQNILLSNPAGR
Lys2
-2.6
10
uM
NPK76-II-72-1 HeLa ULK3
EVVAIkCVAK
Lys1
-26.8
10
uM
NPK76-II-72-1 HeLa Wnk1,Wnk2,Wnk3
DLkCDNIFITGPTGSVK
Lys2
-9.3
10
uM
NPK76-II-72-1 PC-3 Wnk1,Wnk2,Wnk4
IGDLGLATLkR
Activation Loop
-4.5
10
uM
NPK76-II-72-1 PC-3 WNK4
DLkCDNVFITGPTGSVK
Lys2
3.0
10
uM
NPK76-II-72-1 HeLa ZC1/HGK,ZC2/TNIK,ZC3/MINK
DIkGQNVLLTENAEVK
Lys2
-16.4
10
uM
NPK76-II-72-1 PC-3 ZC1/HGK,ZC2/TNIK,ZC3/MINK
DIkGQNVLLTENAEVK
Lys2
-1.9
10
uM