NPK76-II-72-1 KiNativ -- single dose experiment - Dataset (ID:20106)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
NPK76-II-72-1 | PC-3 | SLK | ETSVLAAAkVIDTK | Lys1 | 68.4 | 10 | uM |
NPK76-II-72-1 | HeLa | SLK | DLkAGNILFTLDGDIK | Lys2 | 46.4 | 10 | uM |
NPK76-II-72-1 | PC-3 | SLK | DLkAGNILFTLDGDIK | Lys2 | 12.8 | 10 | uM |
NPK76-II-72-1 | HeLa | SMG1 | DTVTIHSVGGTITILPTkTKPK | ATP | -7.2 | 10 | uM |
NPK76-II-72-1 | PC-3 | SRPK1 | IIHTDIkPENILLSVNEQYIR | Lys2 | 14.4 | 10 | uM |
NPK76-II-72-1 | HeLa | STLK5 | YSVkVLPWLSPEVLQQNLQGYDAK | Activation Loop | 69.5 | 10 | uM |
NPK76-II-72-1 | HeLa | SYK | ISDFGLSkALR | Activation Loop | -12.9 | 10 | uM |
NPK76-II-72-1 | HeLa | TAO1,TAOK3 | DIkAGNILLTEPGQVK | Lys2 | -21.1 | 10 | uM |
NPK76-II-72-1 | PC-3 | TAO1,TAOK3 | DIkAGNILLTEPGQVK | Lys2 | -2.8 | 10 | uM |
NPK76-II-72-1 | PC-3 | TAOK2 | DVkAGNILLSEPGLVK | Lys2 | 1.7 | 10 | uM |
NPK76-II-72-1 | HeLa | TBK1 | TGDLFAIkVFNNISFLRPVDVQMR | Lys1 | 50.3 | 10 | uM |
NPK76-II-72-1 | PC-3 | TLK1 | YAAVkIHQLNK | Lys1 | -9.5 | 10 | uM |
NPK76-II-72-1 | HeLa | TLK1 | YLNEIKPPIIHYDLkPGNILLVDGTACGEIK | Lys2 | 12.6 | 10 | uM |
NPK76-II-72-1 | PC-3 | TLK1 | YLNEIKPPIIHYDLkPGNILLVDGTACGEIK | Lys2 | -19.2 | 10 | uM |
NPK76-II-72-1 | PC-3 | TLK2 | YVAVkIHQLNK | Lys1 | -25.5 | 10 | uM |
NPK76-II-72-1 | HeLa | ULK1 | DLkPQNILLSNPAGR | Lys2 | -2.6 | 10 | uM |
NPK76-II-72-1 | HeLa | ULK3 | EVVAIkCVAK | Lys1 | -26.8 | 10 | uM |
NPK76-II-72-1 | HeLa | Wnk1,Wnk2,Wnk3 | DLkCDNIFITGPTGSVK | Lys2 | -9.3 | 10 | uM |
NPK76-II-72-1 | PC-3 | Wnk1,Wnk2,Wnk4 | IGDLGLATLkR | Activation Loop | -4.5 | 10 | uM |
NPK76-II-72-1 | PC-3 | WNK4 | DLkCDNVFITGPTGSVK | Lys2 | 3.0 | 10 | uM |
NPK76-II-72-1 | HeLa | ZC1/HGK,ZC2/TNIK,ZC3/MINK | DIkGQNVLLTENAEVK | Lys2 | -16.4 | 10 | uM |
NPK76-II-72-1 | PC-3 | ZC1/HGK,ZC2/TNIK,ZC3/MINK | DIkGQNVLLTENAEVK | Lys2 | -1.9 | 10 | uM |