NPK76-II-72-1 KiNativ -- single dose experiment - Dataset (ID:20106)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
NPK76-II-72-1 PC-3 PEK
DLkPSNIFFTMDDVVK
Lys2
52.3
10
uM
NPK76-II-72-1 PC-3 SRPK1
IIHTDIkPENILLSVNEQYIR
Lys2
14.4
10
uM
NPK76-II-72-1 PC-3 PRP4
CNILHADIkPDNILVNESK
Lys2
-31.0
10
uM
NPK76-II-72-1 PC-3 ANPb
GMAFLHNSIISSHGSLkSSNCVVDSR
Lys2
-35.6
10
uM
NPK76-II-72-1 PC-3 CaMK2a,CaMK2b,CaMK2d,CaMK2g
DLkPENLLLASK
Lys2
65.5
10
uM
NPK76-II-72-1 PC-3 CK2a2
DVkPHNVMIDHQQK
Lys2
18.3
10
uM
NPK76-II-72-1 PC-3 MRCKb
DIkPDNVLLDVNGHIR
Lys2
3.2
10
uM
NPK76-II-72-1 HeLa RIPK3
DLkPSNVLLDPELHVK
Lys2
-1.9
10
uM
NPK76-II-72-1 PC-3 MK14
QELNkTIWEVPER
Other
-24.1
10
uM
NPK76-II-72-1 PC-3 MRCKb
NHHVHLYPWSSLDGAEGSFDIkLPETK
Other
-27.0
10
uM
NPK76-II-72-1 HeLa MK14
QELNkTIWEVPER
Other
-19.0
10
uM
NPK76-II-72-1 HeLa JAK1
QLASALSYLEDKDLVHGNVCTkNLLLAR
Other
84.2
10
uM
NPK76-II-72-1 PC-3 MK11
QELNkTVWEVPQR
Other
-46.2
10
uM
NPK76-II-72-1 PC-3 ROCK1
kLQLELNQER
Other
4.4
10
uM
NPK76-II-72-1 PC-3 ILK
ISMADVkFSFQCPGR
Protein Kinase Domain
-3.9
10
uM
NPK76-II-72-1 HeLa eEF2K
YIkYNSNSGFVR
Protein Kinase Domain
-4.9
10
uM
NPK76-II-72-1 PC-3 eEF2K
YIkYNSNSGFVR
Protein Kinase Domain
-16.5
10
uM
NPK76-II-72-1 HeLa KSR1,KSR2
SkNVFYDNGK
Protein Kinase Domain
-26.5
10
uM
NPK76-II-72-1 HeLa RSKL1_domain1
VLGVIDkVLLVMDTR
Protein Kinase Domain
-207.2
10
uM
NPK76-II-72-1 PC-3 RSK2_domain2
SkRDPTEEIEILLR
Protein Kinase Domain
15.9
10
uM
NPK76-II-72-1 HeLa RSK2_domain2
SkRDPTEEIEILLR
Protein Kinase Domain
14.1
10
uM
NPK76-II-72-1 HeLa PAN3
VMDPTkILITGK
-19.2
10
uM