NPK76-II-72-1 KiNativ -- single dose experiment - Dataset (ID:20106)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
NPK76-II-72-1 | PC-3 | PEK | DLkPSNIFFTMDDVVK | Lys2 | 52.3 | 10 | uM |
NPK76-II-72-1 | PC-3 | SRPK1 | IIHTDIkPENILLSVNEQYIR | Lys2 | 14.4 | 10 | uM |
NPK76-II-72-1 | PC-3 | PRP4 | CNILHADIkPDNILVNESK | Lys2 | -31.0 | 10 | uM |
NPK76-II-72-1 | PC-3 | ANPb | GMAFLHNSIISSHGSLkSSNCVVDSR | Lys2 | -35.6 | 10 | uM |
NPK76-II-72-1 | PC-3 | CaMK2a,CaMK2b,CaMK2d,CaMK2g | DLkPENLLLASK | Lys2 | 65.5 | 10 | uM |
NPK76-II-72-1 | PC-3 | CK2a2 | DVkPHNVMIDHQQK | Lys2 | 18.3 | 10 | uM |
NPK76-II-72-1 | PC-3 | MRCKb | DIkPDNVLLDVNGHIR | Lys2 | 3.2 | 10 | uM |
NPK76-II-72-1 | HeLa | RIPK3 | DLkPSNVLLDPELHVK | Lys2 | -1.9 | 10 | uM |
NPK76-II-72-1 | PC-3 | MK14 | QELNkTIWEVPER | Other | -24.1 | 10 | uM |
NPK76-II-72-1 | PC-3 | MRCKb | NHHVHLYPWSSLDGAEGSFDIkLPETK | Other | -27.0 | 10 | uM |
NPK76-II-72-1 | HeLa | MK14 | QELNkTIWEVPER | Other | -19.0 | 10 | uM |
NPK76-II-72-1 | HeLa | JAK1 | QLASALSYLEDKDLVHGNVCTkNLLLAR | Other | 84.2 | 10 | uM |
NPK76-II-72-1 | PC-3 | MK11 | QELNkTVWEVPQR | Other | -46.2 | 10 | uM |
NPK76-II-72-1 | PC-3 | ROCK1 | kLQLELNQER | Other | 4.4 | 10 | uM |
NPK76-II-72-1 | PC-3 | ILK | ISMADVkFSFQCPGR | Protein Kinase Domain | -3.9 | 10 | uM |
NPK76-II-72-1 | HeLa | eEF2K | YIkYNSNSGFVR | Protein Kinase Domain | -4.9 | 10 | uM |
NPK76-II-72-1 | PC-3 | eEF2K | YIkYNSNSGFVR | Protein Kinase Domain | -16.5 | 10 | uM |
NPK76-II-72-1 | HeLa | KSR1,KSR2 | SkNVFYDNGK | Protein Kinase Domain | -26.5 | 10 | uM |
NPK76-II-72-1 | HeLa | RSKL1_domain1 | VLGVIDkVLLVMDTR | Protein Kinase Domain | -207.2 | 10 | uM |
NPK76-II-72-1 | PC-3 | RSK2_domain2 | SkRDPTEEIEILLR | Protein Kinase Domain | 15.9 | 10 | uM |
NPK76-II-72-1 | HeLa | RSK2_domain2 | SkRDPTEEIEILLR | Protein Kinase Domain | 14.1 | 10 | uM |
NPK76-II-72-1 | HeLa | PAN3 | VMDPTkILITGK | -19.2 | 10 | uM |