NPK76-II-72-1 KiNativ -- single dose experiment - Dataset (ID:20106)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
NPK76-II-72-1 HeLa DMPK
DIkPDNILLDR
Lys2
-7.7
10
uM
NPK76-II-72-1 HeLa ABL,ARG
LMTGDTYTAHAGAkFPIK
Activation Loop
-31.1
10
uM
NPK76-II-72-1 HeLa DNAPK
GHDEREHPFLVkGGEDLRQDQR
ATP
-23.8
10
uM
NPK76-II-72-1 HeLa MSK1_domain1
DIkLENILLDSNGHVVLTDFGLSK
Lys2
-0.9
10
uM
NPK76-II-72-1 HeLa eEF2K
YIkYNSNSGFVR
Protein Kinase Domain
-4.9
10
uM
NPK76-II-72-1 HeLa ARAF
DLkSNNIFLHEGLTVK
Lys2
-2.4
10
uM
NPK76-II-72-1 HeLa AMPKa1,AMPKa2
DLkPENVLLDAHMNAK
Lys2
-14.5
10
uM
NPK76-II-72-1 HeLa CDK2
DLkPQNLLINTEGAIK
Lys2
0.5
10
uM
NPK76-II-72-1 HeLa MK03
DLkPSNLLINTTCDLK
Lys2
7.7
10
uM
NPK76-II-72-1 HeLa ATR
FYIMMCkPK
ATP
-80.8
10
uM
NPK76-II-72-1 HeLa Erk5
DLkPSNLLVNENCELK
Lys2
22.6
10
uM
NPK76-II-72-1 HeLa JAK1_domain2
IGDFGLTkAIETDKEYYTVK
Activation Loop
-25.1
10
uM
NPK76-II-72-1 HeLa FER
TSVAVkTCKEDLPQELK
Lys1
16.4
10
uM
NPK76-II-72-1 HeLa CDK7
DLkPNNLLLDENGVLK
Lys2
-6.7
10
uM
NPK76-II-72-1 HeLa LOK
DLkAGNVLMTLEGDIR
Lys2
7.9
10
uM
NPK76-II-72-1 HeLa GCK
DTVTSELAAVkIVK
Lys1
3.2
10
uM
NPK76-II-72-1 HeLa ACK
TVSVAVkCLKPDVLSQPEAMDDFIR
Lys1
-1.0
10
uM
NPK76-II-72-1 HeLa GSK3A
DIkPQNLLVDPDTAVLK
Lys2
-3.8
10
uM
NPK76-II-72-1 HeLa BRAF
DLkSNNIFLHEDLTVK
Lys2
-6.5
10
uM
NPK76-II-72-1 HeLa IKKA
DLkPENIVLQDVGGK
Lys2
-14.5
10
uM
NPK76-II-72-1 HeLa IKKE,TBK1
DIkPGNIMR
Lys2
-18.4
10
uM
NPK76-II-72-1 HeLa CaMK1a
LVAIkCIAK
Lys1
10.8
10
uM
NPK76-II-72-1 HeLa AMPKa1,AMPKa2
VAVkILNR
Lys1
-30.6
10
uM
NPK76-II-72-1 HeLa NEK1
DIkSQNIFLTK
Lys2
-0.3
10
uM
NPK76-II-72-1 HeLa ILK
WQGNDIVVkVLK
Lys1
-4.3
10
uM