NPK76-II-72-1 KiNativ -- single dose experiment - Dataset (ID:20106)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| NPK76-II-72-1 | PC-3 | CSK | VSDFGLTkEASSTQDTGKLPVK | Activation Loop | -11.0 | 10 | uM |
| NPK76-II-72-1 | HeLa | DMPK | DIkPDNILLDR | Lys2 | -7.7 | 10 | uM |
| NPK76-II-72-1 | PC-3 | DNAPK | kGGSWIQEINVAEK | ATP | 24.9 | 10 | uM |
| NPK76-II-72-1 | HeLa | DNAPK | GHDEREHPFLVkGGEDLRQDQR | ATP | -23.8 | 10 | uM |
| NPK76-II-72-1 | PC-3 | DNAPK | GHDEREHPFLVkGGEDLRQDQR | ATP | -22.7 | 10 | uM |
| NPK76-II-72-1 | HeLa | eEF2K | YIkYNSNSGFVR | Protein Kinase Domain | -4.9 | 10 | uM |
| NPK76-II-72-1 | PC-3 | eEF2K | YIkYNSNSGFVR | Protein Kinase Domain | -16.5 | 10 | uM |
| NPK76-II-72-1 | PC-3 | EGFR | IPVAIkELR | Lys1 | 10.7 | 10 | uM |
| NPK76-II-72-1 | PC-3 | EPHA2 | VLEDDPEATYTTSGGkIPIR | Activation Loop | -2.8 | 10 | uM |
| NPK76-II-72-1 | HeLa | MK03 | DLkPSNLLINTTCDLK | Lys2 | 7.7 | 10 | uM |
| NPK76-II-72-1 | PC-3 | MK03 | DLkPSNLLINTTCDLK | Lys2 | -1.2 | 10 | uM |
| NPK76-II-72-1 | HeLa | Erk5 | DLkPSNLLVNENCELK | Lys2 | 22.6 | 10 | uM |
| NPK76-II-72-1 | PC-3 | FAK | CIGEGQFGDVHQGIYMSPENPALAVAIkTCK | Lys1 | 90.1 | 10 | uM |
| NPK76-II-72-1 | HeLa | FER | TSVAVkTCKEDLPQELK | Lys1 | 16.4 | 10 | uM |
| NPK76-II-72-1 | PC-3 | FER | TSVAVkTCKEDLPQELK | Lys1 | 43.3 | 10 | uM |
| NPK76-II-72-1 | PC-3 | FYN,SRC,YES | QGAkFPIKWTAPEAALYGR | Activation Loop | -44.1 | 10 | uM |
| NPK76-II-72-1 | HeLa | GCK | DTVTSELAAVkIVK | Lys1 | 3.2 | 10 | uM |
| NPK76-II-72-1 | PC-3 | GCN2_domain2 | DLkPVNIFLDSDDHVK | Lys2 | -4.0 | 10 | uM |
| NPK76-II-72-1 | HeLa | GSK3A | DIkPQNLLVDPDTAVLK | Lys2 | -3.8 | 10 | uM |
| NPK76-II-72-1 | PC-3 | GSK3B | DIkPQNLLLDPDTAVLK | Lys2 | -7.0 | 10 | uM |
| NPK76-II-72-1 | HeLa | IKKA | DLkPENIVLQDVGGK | Lys2 | -14.5 | 10 | uM |
| NPK76-II-72-1 | HeLa | IKKE,TBK1 | DIkPGNIMR | Lys2 | -18.4 | 10 | uM |
| NPK76-II-72-1 | PC-3 | IKKE,TBK1 | DIkPGNIMR | Lys2 | 12.4 | 10 | uM |
| NPK76-II-72-1 | PC-3 | ILK | ISMADVkFSFQCPGR | Protein Kinase Domain | -3.9 | 10 | uM |
| NPK76-II-72-1 | HeLa | ILK | WQGNDIVVkVLK | Lys1 | -4.3 | 10 | uM |