CH5424802 KiNativ -- single dose experiment - Dataset (ID:20105)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
CH5424802 HeLa RSK1 domain1
DLKPENILLDEEGHIkLTDFGLSKEAIDHEK
Lys2
76.9
10
uM
CH5424802 HeLa MK14
QELNkTIWEVPER
Other
-13.5
10
uM
CH5424802 HeLa CHK1
LSkGDGLEFK
Other
7.5
10
uM
CH5424802 HeLa ROCK1
kLQLELNQER
Other
9.4
10
uM
CH5424802 HeLa PRP4
AAGIGkDFKENPNLR
Other
-19.5
10
uM
CH5424802 HeLa JAK1
QLASALSYLEDKDLVHGNVCTkNLLLAR
Protein Kinase Domain
11.8
10
uM
CH5424802 HeLa ILK
ISMADVkFSFQCPGR
Protein Kinase Domain
-3.5
10
uM
CH5424802 HeLa RSK2_domain2
SkRDPTEEIEILLR
Protein Kinase Domain
60.4
10
uM
CH5424802 HeLa ATR
kAGHHQTAYNALLNAGESR
Protein Kinase Domain
-18.3
10
uM
CH5424802 HeLa RSKL1_domain1
VLGVIDkVLLVMDTR
Protein Kinase Domain
3.9
10
uM