CH5424802 KiNativ -- single dose experiment - Dataset (ID:20105)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| CH5424802 | HeLa | MAP2K3 | MCDFGISGYLVDSVAkTMDAGCKPYMAPER | Activation Loop | 5.2 | 10 | uM |
| CH5424802 | HeLa | PKR | IGDFGLVTSLkNDGKR | Activation Loop | 11.8 | 10 | uM |
| CH5424802 | HeLa | RSK2_domain1 | LTDFGLSkESIDHEKK | Activation Loop | 81.3 | 10 | uM |
| CH5424802 | HeLa | JAK1 domain2 | IGDFGLTkAIETDKEYYTVKDDR | Activation Loop | 19.5 | 10 | uM |
| CH5424802 | HeLa | EPHA2 | VLEDDPEATYTTSGGkIPIR | Activation Loop | 19.6 | 10 | uM |
| CH5424802 | HeLa | KS6B1 | LTDFGLCkESIHDGTVTHTFCGTIEYMAPEILMR | Activation Loop | -41.3 | 10 | uM |
| CH5424802 | HeLa | FYN,SRC,YES | QGAkFPIKWTAPEAALYGR | Activation Loop | 18.2 | 10 | uM |
| CH5424802 | HeLa | RSK1_domain1 | LTDFGLSkEAIDHEKK | Activation Loop | 87.9 | 10 | uM |
| CH5424802 | HeLa | EPHB4 | FLEENSSDPTYTSSLGGkIPIR | Activation Loop | 86.0 | 10 | uM |
| CH5424802 | HeLa | EGFR | LLGAEEKEYHAEGGkVPIK | Activation Loop | 12.2 | 10 | uM |
| CH5424802 | HeLa | EGFR | LLGAEEKEYHAEGGkVPIKWMALESILHR | Activation Loop | 3.4 | 10 | uM |
| CH5424802 | HeLa | MAP2K6 | MCDFGISGYLVDSVAkTIDAGCKPYMAPER | Activation Loop | 4.4 | 10 | uM |
| CH5424802 | HeLa | MST3,MST4,YSK1 | LADFGVAGQLTDTQIkR | Activation Loop | 9.5 | 10 | uM |
| CH5424802 | HeLa | NDR1,NDR2 | LSDFGLCTGLkK | Activation Loop | -11.8 | 10 | uM |
| CH5424802 | HeLa | ABL,ARG | LMTGDTYTAHAGAkFPIK | Activation Loop | -2.6 | 10 | uM |
| CH5424802 | HeLa | CSK | VSDFGLTkEASSTQDTGKLPVK | Activation Loop | 1.9 | 10 | uM |
| CH5424802 | HeLa | FER | QEDGGVYSSSGLkQIPIKWTAPEALNYGR | Activation Loop | 95.1 | 10 | uM |
| CH5424802 | HeLa | JAK1_domain2 | IGDFGLTkAIETDKEYYTVK | Activation Loop | -16.3 | 10 | uM |
| CH5424802 | HeLa | Wnk1,Wnk2,Wnk4 | IGDLGLATLkR | Activation Loop | 1.2 | 10 | uM |
| CH5424802 | HeLa | CSK | VSDFGLTkEASSTQDTGKLPVKWTAPEALR | Activation Loop | 13.0 | 10 | uM |
| CH5424802 | HeLa | MET | DMYDkEYYSVHNK | Activation Loop | -5.0 | 10 | uM |
| CH5424802 | HeLa | PIK3C3 | TEDGGkYPVIFKHGDDLR | ATP | 12.2 | 10 | uM |
| CH5424802 | HeLa | PIK3CA | RPLWLNWENPDIMSELLFQNNEIIFkNGDDLRQDMLTLQIIR | ATP | 34.5 | 10 | uM |
| CH5424802 | HeLa | PIK3CB | VFGEDSVGVIFkNGDDLRQDMLTLQMLR | ATP | -8.7 | 10 | uM |
| CH5424802 | HeLa | DNAPK | kGGSWIQEINVAEK | ATP | -19.7 | 10 | uM |