NVP-BHG712 KiNativ -- multiple dose experiment - Dataset (ID:20104)

Proteins Studied

LINCS ID Name HMS LINCS ID UniProt ID Alternative Names Provider Mutation Phosphlorylation State Domain Protein Description
200675 DNAPK 200675 P78527
DNA-dependent protein kinase catalytic subunit
KiNativ
200677 eEF2K 200677 O00418
Elongation factor 2 kinase
KiNativ
200678 EGFR 200678 P00533
Epidermal growth factor receptor precursor
KiNativ
200679 EPHA2 200679 P29317
Ephrin type-A receptor 2
KiNativ
200680 MK03 200680 P27361
Mitogen-activated protein kinase 3
KiNativ
200649 KCC2D 200649 Q13557
Calcium/calmodulin-dependent protein kinase type II subunit delta; CaM kinase II subunit delta; CAMK2D; CAMKD; DKFZp686G23119; DKFZp686I2288; MGC44911
KiNativ
200636 AGK 200636 Q53H12
Acylglycerol kinase, mitochondrial
KiNativ
200771 NEK8 200771 Q86SG6
Serine/threonine-protein kinase Nek8
KiNativ
200666 CHK2 200666 O96017
Serine/threonine-protein kinase Chk2; CHK2 checkpoint homolog
KiNativ
200664 CDK9 200664 P50750
Cyclin-dependent kinase 9; cell division protein kinase 9; C-2k; CDC2L4; CDK9; CTK1; PITALRE; TAK
KiNativ
200648 CaMK1a 200648 Q14012
Calcium/calmodulin-dependent protein kinase I; CAMK1; CaMK1a; CAMKI; MGC120317; MGC120318
KiNativ
200663 CDK7 200663 P50613
Cyclin-dependent kinase 7; cell division protein kinase 7; CAK1; CDK7; CDKN7; MO15; p39MO15; STK1
KiNativ
200693 GSK3A 200693 P49840
Glycogen synthase kinase-3 alpha
KiNativ
200661 CDK5 200661 Q00535
Cyclin-dependent kinase 5; cell division protein kinase 5; PSSALRE
KiNativ
200647 BRAF 200647 P15056
Serine/threonine-protein kinase B-raf; v-raf murine sarcoma viral oncogene homolog B1; BRAF1; RAFB1
KiNativ
200694 GSK3B 200694 P49841
Glycogen synthase kinase-3 beta
KiNativ
200695 IKKA 200695 O15111
Inhibitor of nuclear factor kappa-B kinase subunit alpha
KiNativ
200696 IKKB 200696 O14920
Inhibitor of nuclear factor kappa-B kinase subunit beta
KiNativ
200697 IKKE,TBK1 200697 Q14164
Inhibitor of nuclear factor kappa-B kinase subunit epsilon
KiNativ
200698 ILK 200698 Q13418
Integrin-linked protein kinase 1
KiNativ
200699 ILK 200699 Q13418
Integrin-linked protein kinase 1
KiNativ
200700 IRAK1 200700 P51617
Interleukin-1 receptor-associated kinase 1
KiNativ
200701 IRAK4 200701 Q9NWZ3
Interleukin-1 receptor-associated kinase 4; IPD1; NY-REN-64; REN64
KiNativ
200635 ACK 200635 Q07912
Activated CDC42 kinase 1
KiNativ
200690 GCK 200690 Q12851
Mitogen-activated protein kinase kinase kinase kinase 2
KiNativ