NVP-BHG712 KiNativ -- multiple dose experiment - Dataset (ID:20104)

Proteins Studied

LINCS ID Name HMS LINCS ID UniProt ID Alternative Names Provider Mutation Phosphlorylation State Domain Protein Description
201091 CDK14 201091 O94921
Cyclin-dependent kinase 14; serine/threonine-protein kinase PFTAIRE-1; PFTK1
KiNativ
200783 CDK16 200783 Q00536
Cyclin-dependent kinase 16; Cell division protein kinase 16; Serine/threonine-protein kinase PCTAIRE-1; FLJ16665; PCTAIRE; PCTAIRE1; PCTGAIRE; PCTK1
KiNativ
201082 CDK2 201082 P24941
Cyclin-dependent kinase 2; p33 protein kinase
KiNativ
200657 CDK2 200657 P24941
Cyclin-dependent kinase 2; p33 protein kinase
KiNativ
200658 CDK2 200658 P24941
Cyclin-dependent kinase 2; p33 protein kinase
KiNativ
200661 CDK5 200661 Q00535
Cyclin-dependent kinase 5; cell division protein kinase 5; PSSALRE
KiNativ
200890 CDK5 200890 Q00535
Cyclin-dependent kinase 5; cell division protein kinase 5; PSSALRE
KiNativ
201048 CDK5 201048 Q00535
Cyclin-dependent kinase 5; cell division protein kinase 5; PSSALRE
KiNativ
200663 CDK7 200663 P50613
Cyclin-dependent kinase 7; cell division protein kinase 7; CAK1; CDK7; CDKN7; MO15; p39MO15; STK1
KiNativ
200664 CDK9 200664 P50750
Cyclin-dependent kinase 9; cell division protein kinase 9; C-2k; CDC2L4; CDK9; CTK1; PITALRE; TAK
KiNativ
200894 CHK1 200894 O14757
Serine/threonine-protein kinase Chk1; CHK1 checkpoint homolog
KiNativ
200896 CHK2 200896 O96017
Serine/threonine-protein kinase Chk2; CHK2 checkpoint homolog
KiNativ
200666 CHK2 200666 O96017
Serine/threonine-protein kinase Chk2; CHK2 checkpoint homolog
KiNativ
200905 CSK 200905 P41240
Tyrosine-protein kinase CSK
KiNativ
200669 CSK 200669 P41240
Tyrosine-protein kinase CSK
KiNativ
201083 DGKH 201083 Q86XP1
Diacylglycerol kinase eta2
KiNativ
200675 DNAPK 200675 P78527
DNA-dependent protein kinase catalytic subunit
KiNativ
200672 DNAPK 200672 P78527
DNA-dependent protein kinase catalytic subunit
KiNativ
200677 eEF2K 200677 O00418
Elongation factor 2 kinase
KiNativ
200678 EGFR 200678 P00533
Epidermal growth factor receptor precursor
KiNativ
201035 EGFR 201035 P00533
Epidermal growth factor receptor precursor
KiNativ
201050 EGFR 201050 P00533
Epidermal growth factor receptor precursor
KiNativ
201051 EphA1 201051 P21709
Ephrin type-A receptor 1 precursor
KiNativ
200679 EPHA2 200679 P29317
Ephrin type-A receptor 2
KiNativ
201052 EPHA2 201052 P29317
Ephrin type-A receptor 2
KiNativ