NVP-BHG712 KiNativ -- multiple dose experiment - Dataset (ID:20104)

Proteins Studied

LINCS ID Name HMS LINCS ID UniProt ID Alternative Names Provider Mutation Phosphlorylation State Domain Protein Description
200675 DNAPK 200675 P78527
DNA-dependent protein kinase catalytic subunit
KiNativ
200677 eEF2K 200677 O00418
Elongation factor 2 kinase
KiNativ
200678 EGFR 200678 P00533
Epidermal growth factor receptor precursor
KiNativ
200679 EPHA2 200679 P29317
Ephrin type-A receptor 2
KiNativ
200680 MK03 200680 P27361
Mitogen-activated protein kinase 3
KiNativ
200681 MK03 200681 P27361
Mitogen-activated protein kinase 3
KiNativ
200682 Erk5 200682 Q13164
Mitogen-activated protein kinase 7
KiNativ
200683 FAK 200683 Q05397
Focal adhesion kinase 1
KiNativ
200686 FER 200686 P16591
Proto-oncogene tyrosine-protein kinase FER
KiNativ
200687 FYN,SRC,YES 200687 P06241
Proto-oncogene tyrosine-protein kinase Fyn
KiNativ
200689 GCK 200689 Q12851
Mitogen-activated protein kinase kinase kinase kinase 2
KiNativ
200690 GCK 200690 Q12851
Mitogen-activated protein kinase kinase kinase kinase 2
KiNativ
200691 GCN2_domain2 200691 Q9P2K8
Eukaryotic translation initiation factor 2-alpha kinase 4
KiNativ domain2
200692 GCN2_domain2 200692 Q9P2K8
Eukaryotic translation initiation factor 2-alpha kinase 4
KiNativ domain2
200693 GSK3A 200693 P49840
Glycogen synthase kinase-3 alpha
KiNativ
200694 GSK3B 200694 P49841
Glycogen synthase kinase-3 beta
KiNativ
200695 IKKA 200695 O15111
Inhibitor of nuclear factor kappa-B kinase subunit alpha
KiNativ
200696 IKKB 200696 O14920
Inhibitor of nuclear factor kappa-B kinase subunit beta
KiNativ
200697 IKKE,TBK1 200697 Q14164
Inhibitor of nuclear factor kappa-B kinase subunit epsilon
KiNativ
200698 ILK 200698 Q13418
Integrin-linked protein kinase 1
KiNativ
200699 ILK 200699 Q13418
Integrin-linked protein kinase 1
KiNativ
200700 IRAK1 200700 P51617
Interleukin-1 receptor-associated kinase 1
KiNativ
200701 IRAK4 200701 Q9NWZ3
Interleukin-1 receptor-associated kinase 4; IPD1; NY-REN-64; REN64
KiNativ
200702 IRE1 200702 O75460
Serine/threonine-protein kinase/endoribonuclease IRE1
KiNativ
200703 ITPK1 200703 Q13572
Inositol-tetrakisphosphate 1-kinase
KiNativ