XMD-12 KiNativ -- single dose experiment - Dataset (ID:20103)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
XMD-12 | PC-3 | EGFR | IPVAIkELR | Lys1 | -0.3 | 10 | uM |
XMD-12 | PC-3 | EphA1 | LLDDFDGTYETQGGkIPIR | Activation Loop | 46.7 | 10 | uM |
XMD-12 | PC-3 | EPHA2 | EVPVAIkTLK | Lys1 | 8.4 | 10 | uM |
XMD-12 | PC-3 | EPHA2 | VLEDDPEATYTTSGGkIPIR | Activation Loop | 2.2 | 10 | uM |
XMD-12 | PC-3 | EphA7 | VIEDDPEAVYTTTGGkIPVR | Activation Loop | -21.4 | 10 | uM |
XMD-12 | PC-3 | EPHB2 | FLEDDTSDPTYTSALGGkIPIR | Activation Loop | 27.3 | 10 | uM |
XMD-12 | PC-3 | EPHB4 | FLEENSSDPTYTSSLGGkIPIR | Activation Loop | 51.7 | 10 | uM |
XMD-12 | HeLa | Erk5 | DLkPSNLLVNENCELK | Lys2 | 97.4 | 10 | uM |
XMD-12 | PC-3 | FAK | CIGEGQFGDVHQGIYMSPENPALAVAIkTCK | Lys1 | 85.4 | 10 | uM |
XMD-12 | PC-3 | FER | TSVAVkTCKEDLPQELK | Lys1 | 42.4 | 10 | uM |
XMD-12 | HeLa | FER | TSVAVkTCKEDLPQELK | Lys1 | 30.6 | 10 | uM |
XMD-12 | HeLa | FES | LRADNTLVAVkSCR | Lys1 | -2.5 | 10 | uM |
XMD-12 | PC-3 | FYN,SRC,YES | QGAkFPIKWTAPEAALYGR | Activation Loop | 70.5 | 10 | uM |
XMD-12 | HeLa | GCK | DTVTSELAAVkIVK | Lys1 | 15.0 | 10 | uM |
XMD-12 | PC-3 | GCN2 | LDGCCYAVkR | Lys1 | -12.4 | 10 | uM |
XMD-12 | HeLa | GCN2 | LDGCCYAVkR | Lys1 | -5.1 | 10 | uM |
XMD-12 | PC-3 | GCN2_domain2 | DLkPVNIFLDSDDHVK | Lys2 | 0.2 | 10 | uM |
XMD-12 | HeLa | GSK3A | DIkPQNLLVDPDTAVLK | Lys2 | -16.7 | 10 | uM |
XMD-12 | PC-3 | GSK3B | DIkPQNLLLDPDTAVLK | Lys2 | 2.9 | 10 | uM |
XMD-12 | HeLa | HPK1 | DKVSGDLVALkMVK | Lys1 | 69.0 | 10 | uM |
XMD-12 | HeLa | IKKA | DLkPENIVLQDVGGK | Lys2 | -7.3 | 10 | uM |
XMD-12 | HeLa | IKKE | SGELVAVkVFNTTSYLRPR | Lys1 | 14.6 | 10 | uM |
XMD-12 | PC-3 | IKKE,TBK1 | DIkPGNIMR | Lys2 | 64.7 | 10 | uM |
XMD-12 | HeLa | IKKE,TBK1 | DIkPGNIMR | Lys2 | 24.9 | 10 | uM |
XMD-12 | PC-3 | ILK | ISMADVkFSFQCPGR | Protein Kinase Domain | -11.9 | 10 | uM |