XMD-12 KiNativ -- single dose experiment - Dataset (ID:20103)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD-12 PC-3 EGFR
IPVAIkELR
Lys1
-0.3
10
uM
XMD-12 PC-3 EphA1
LLDDFDGTYETQGGkIPIR
Activation Loop
46.7
10
uM
XMD-12 PC-3 EPHA2
EVPVAIkTLK
Lys1
8.4
10
uM
XMD-12 PC-3 EPHA2
VLEDDPEATYTTSGGkIPIR
Activation Loop
2.2
10
uM
XMD-12 PC-3 EphA7
VIEDDPEAVYTTTGGkIPVR
Activation Loop
-21.4
10
uM
XMD-12 PC-3 EPHB2
FLEDDTSDPTYTSALGGkIPIR
Activation Loop
27.3
10
uM
XMD-12 PC-3 EPHB4
FLEENSSDPTYTSSLGGkIPIR
Activation Loop
51.7
10
uM
XMD-12 HeLa Erk5
DLkPSNLLVNENCELK
Lys2
97.4
10
uM
XMD-12 PC-3 FAK
CIGEGQFGDVHQGIYMSPENPALAVAIkTCK
Lys1
85.4
10
uM
XMD-12 PC-3 FER
TSVAVkTCKEDLPQELK
Lys1
42.4
10
uM
XMD-12 HeLa FER
TSVAVkTCKEDLPQELK
Lys1
30.6
10
uM
XMD-12 HeLa FES
LRADNTLVAVkSCR
Lys1
-2.5
10
uM
XMD-12 PC-3 FYN,SRC,YES
QGAkFPIKWTAPEAALYGR
Activation Loop
70.5
10
uM
XMD-12 HeLa GCK
DTVTSELAAVkIVK
Lys1
15.0
10
uM
XMD-12 PC-3 GCN2
LDGCCYAVkR
Lys1
-12.4
10
uM
XMD-12 HeLa GCN2
LDGCCYAVkR
Lys1
-5.1
10
uM
XMD-12 PC-3 GCN2_domain2
DLkPVNIFLDSDDHVK
Lys2
0.2
10
uM
XMD-12 HeLa GSK3A
DIkPQNLLVDPDTAVLK
Lys2
-16.7
10
uM
XMD-12 PC-3 GSK3B
DIkPQNLLLDPDTAVLK
Lys2
2.9
10
uM
XMD-12 HeLa HPK1
DKVSGDLVALkMVK
Lys1
69.0
10
uM
XMD-12 HeLa IKKA
DLkPENIVLQDVGGK
Lys2
-7.3
10
uM
XMD-12 HeLa IKKE
SGELVAVkVFNTTSYLRPR
Lys1
14.6
10
uM
XMD-12 PC-3 IKKE,TBK1
DIkPGNIMR
Lys2
64.7
10
uM
XMD-12 HeLa IKKE,TBK1
DIkPGNIMR
Lys2
24.9
10
uM
XMD-12 PC-3 ILK
ISMADVkFSFQCPGR
Protein Kinase Domain
-11.9
10
uM