XMD-12 KiNativ -- single dose experiment - Dataset (ID:20103)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
XMD-12 | HeLa | TBK1 | TGDLFAIkVFNNISFLRPVDVQMR | Lys1 | 10 | uM | |
XMD-12 | PC-3 | PI42C | TLVIkEVSSEDIADMHSNLSNYHQYIVK | ATP | 76.2 | 10 | uM |
XMD-12 | HeLa | PI42C | TLVIkEVSSEDIADMHSNLSNYHQYIVK | ATP | 60.5 | 10 | uM |
XMD-12 | PC-3 | CaMK2g | TSTQEYAAkIINTK | Lys1 | 33.0 | 10 | uM |
XMD-12 | HeLa | CaMK2g | TSTQEYAAkIINTK | Lys1 | 19.3 | 10 | uM |
XMD-12 | HeLa | FER | TSVAVkTCKEDLPQELK | Lys1 | 30.6 | 10 | uM |
XMD-12 | PC-3 | FER | TSVAVkTCKEDLPQELK | Lys1 | 42.4 | 10 | uM |
XMD-12 | HeLa | ACK | TVSVAVkCLKPDVLSQPEAMDDFIR | Lys1 | 87.9 | 10 | uM |
XMD-12 | PC-3 | CHK2 | VAIkIISK | Lys1 | 22.9 | 10 | uM |
XMD-12 | PC-3 | SRC | VAIkTLKPGTMSPEAFLQEAQVMK | Lys1 | 94.6 | 10 | uM |
XMD-12 | HeLa | AMPKa1,AMPKa2 | VAVkILNR | Lys1 | 88.7 | 10 | uM |
XMD-12 | PC-3 | AMPKa1,AMPKa2 | VAVkILNR | Lys1 | 90.3 | 10 | uM |
XMD-12 | HeLa | LYN | VAVkTLKPGTMSVQAFLEEANLMK | Lys1 | 51.7 | 10 | uM |
XMD-12 | HeLa | LATS2 | VDTHALYAMkTLR | Lys1 | -22.6 | 10 | uM |
XMD-12 | PC-3 | PIK3CB | VFGEDSVGVIFkNGDDLRQDMLTLQMLR | ATP | -25.3 | 10 | uM |
XMD-12 | PC-3 | EphA7 | VIEDDPEAVYTTTGGkIPVR | Activation Loop | -21.4 | 10 | uM |
XMD-12 | PC-3 | EPHA2 | VLEDDPEATYTTSGGkIPIR | Activation Loop | 2.2 | 10 | uM |
XMD-12 | HeLa | RSK1,RSK4 domain1 | VLGQGSFGkVFLVR | ATP Loop | -11.2 | 10 | uM |
XMD-12 | HeLa | MSK1,MSK2_domain1 | VLGTGAYGkVFLVR | ATP Loop | 14.4 | 10 | uM |
XMD-12 | HeLa | RSKL1_domain1 | VLGVIDkVLLVMDTR | Protein Kinase Domain | -23.2 | 10 | uM |
XMD-12 | HeLa | PAN3 | VMDPTkILITGK | -13.7 | 10 | uM | |
XMD-12 | HeLa | PI4KB | VPHTQAVVLNSkDK | ATP | -5.8 | 10 | uM |
XMD-12 | PC-3 | PI4KB | VPHTQAVVLNSkDK | ATP | 0.2 | 10 | uM |
XMD-12 | PC-3 | CSK | VSDFGLTkEASSTQDTGKLPVK | Activation Loop | -23.4 | 10 | uM |
XMD-12 | HeLa | CSK | VSDFGLTkEASSTQDTGKLPVK | Activation Loop | -14.1 | 10 | uM |