XMD-12 KiNativ -- single dose experiment - Dataset (ID:20103)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD-12 HeLa TBK1
TGDLFAIkVFNNISFLRPVDVQMR
Lys1
10
uM
XMD-12 PC-3 PI42C
TLVIkEVSSEDIADMHSNLSNYHQYIVK
ATP
76.2
10
uM
XMD-12 HeLa PI42C
TLVIkEVSSEDIADMHSNLSNYHQYIVK
ATP
60.5
10
uM
XMD-12 PC-3 CaMK2g
TSTQEYAAkIINTK
Lys1
33.0
10
uM
XMD-12 HeLa CaMK2g
TSTQEYAAkIINTK
Lys1
19.3
10
uM
XMD-12 HeLa FER
TSVAVkTCKEDLPQELK
Lys1
30.6
10
uM
XMD-12 PC-3 FER
TSVAVkTCKEDLPQELK
Lys1
42.4
10
uM
XMD-12 HeLa ACK
TVSVAVkCLKPDVLSQPEAMDDFIR
Lys1
87.9
10
uM
XMD-12 PC-3 CHK2
VAIkIISK
Lys1
22.9
10
uM
XMD-12 PC-3 SRC
VAIkTLKPGTMSPEAFLQEAQVMK
Lys1
94.6
10
uM
XMD-12 HeLa AMPKa1,AMPKa2
VAVkILNR
Lys1
88.7
10
uM
XMD-12 PC-3 AMPKa1,AMPKa2
VAVkILNR
Lys1
90.3
10
uM
XMD-12 HeLa LYN
VAVkTLKPGTMSVQAFLEEANLMK
Lys1
51.7
10
uM
XMD-12 HeLa LATS2
VDTHALYAMkTLR
Lys1
-22.6
10
uM
XMD-12 PC-3 PIK3CB
VFGEDSVGVIFkNGDDLRQDMLTLQMLR
ATP
-25.3
10
uM
XMD-12 PC-3 EphA7
VIEDDPEAVYTTTGGkIPVR
Activation Loop
-21.4
10
uM
XMD-12 PC-3 EPHA2
VLEDDPEATYTTSGGkIPIR
Activation Loop
2.2
10
uM
XMD-12 HeLa RSK1,RSK4 domain1
VLGQGSFGkVFLVR
ATP Loop
-11.2
10
uM
XMD-12 HeLa MSK1,MSK2_domain1
VLGTGAYGkVFLVR
ATP Loop
14.4
10
uM
XMD-12 HeLa RSKL1_domain1
VLGVIDkVLLVMDTR
Protein Kinase Domain
-23.2
10
uM
XMD-12 HeLa PAN3
VMDPTkILITGK
-13.7
10
uM
XMD-12 HeLa PI4KB
VPHTQAVVLNSkDK
ATP
-5.8
10
uM
XMD-12 PC-3 PI4KB
VPHTQAVVLNSkDK
ATP
0.2
10
uM
XMD-12 PC-3 CSK
VSDFGLTkEASSTQDTGKLPVK
Activation Loop
-23.4
10
uM
XMD-12 HeLa CSK
VSDFGLTkEASSTQDTGKLPVK
Activation Loop
-14.1
10
uM