XMD-12 KiNativ -- single dose experiment - Dataset (ID:20103)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD-12 PC-3 M3K2
VYLCYDVDTGRELAVkQVQFDPDSPETSKEVNALECEIQLLK
Lys1
66.5
10
uM
XMD-12 HeLa MLTK
WISQDKEVAVKk
Lys1
11.4
10
uM
XMD-12 PC-3 MLTK
WISQDKEVAVKk
Lys1
15.8
10
uM
XMD-12 PC-3 ILK
WQGIVVkVLK
Lys1
-12.5
10
uM
XMD-12 HeLa ILK
WQGIVVkVLK
Lys1
-4.0
10
uM
XMD-12 HeLa TLK1
YAAVkIHQLNK
Lys1
-23.8
10
uM
XMD-12 PC-3 TLK1
YAAVkIHQLNK
Lys1
-47.5
10
uM
XMD-12 HeLa JAK1_domain2
YDPEGDNTGEQVAVkSLKPESGGNHIADLKK
Lys1
-208.2
10
uM
XMD-12 HeLa WEE1
YIHSMSLVHMDIkPSNIFISR
Lys2
10
uM
XMD-12 HeLa eEF2K
YIkYNSNSGFVR
Protein Kinase Domain
-9.2
10
uM
XMD-12 PC-3 eEF2K
YIkYNSNSGFVR
Protein Kinase Domain
-2.6
10
uM
XMD-12 PC-3 TLK1
YLNEIKPPIIHYDLkPGNILLVDGTACGEIK
Lys2
-7.5
10
uM
XMD-12 HeLa TLK1
YLNEIKPPIIHYDLkPGNILLVDGTACGEIK
Lys2
-20.1
10
uM
XMD-12 HeLa STLK5
YSVkVLPWLSPEVLQQNLQGYDAK
Activation Loop
10
uM
XMD-12 PC-3 TLK2
YVAVkIHQLNK
Lys1
-11.7
10
uM
XMD-12 HeLa TEC
YVLDDQYTSSSGAkFPVK
Activation Loop
11.2
10
uM