XMD-12 KiNativ -- single dose experiment - Dataset (ID:20103)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD-12 HeLa MST3
DIkAANVLLSEHGEVK
Lys2
15.0
10
uM
XMD-12 HeLa JAK1
QLASALSYLEDKDLVHGNVCTkNLLLAR
Other
92.9
10
uM
XMD-12 PC-3 MK11
QELNkTVWEVPQR
Other
31.8
10
uM
XMD-12 PC-3 MRCKb
NHHVHLYPWSSLDGAEGSFDIkLPETK
Other
2.8
10
uM
XMD-12 PC-3 ROCK1
kLQLELNQER
Other
-25.8
10
uM
XMD-12 HeLa MK14
QELNkTIWEVPER
Other
-2.7
10
uM
XMD-12 PC-3 MK14
QELNkTIWEVPER
Other
-5.0
10
uM
XMD-12 HeLa IRAK3
SHLEHQSCTINMTSSSSkHLWYMPEEYIR
Protein Kinase Domain
23.7
10
uM
XMD-12 HeLa eEF2K
YIkYNSNSGFVR
Protein Kinase Domain
-9.2
10
uM
XMD-12 HeLa KSR1,KSR2
SkNVFYDNGK
Protein Kinase Domain
-2.4
10
uM
XMD-12 PC-3 eEF2K
YIkYNSNSGFVR
Protein Kinase Domain
-2.6
10
uM
XMD-12 PC-3 ILK
ISMADVkFSFQCPGR
Protein Kinase Domain
-11.9
10
uM
XMD-12 HeLa RSK2_domain2
SkRDPTEEIEILLR
Protein Kinase Domain
14.8
10
uM
XMD-12 PC-3 RSK2_domain2
SkRDPTEEIEILLR
Protein Kinase Domain
49.7
10
uM
XMD-12 HeLa RSKL1_domain1
VLGVIDkVLLVMDTR
Protein Kinase Domain
-23.2
10
uM
XMD-12 HeLa PAN3
VMDPTkILITGK
-13.7
10
uM