XMD-12 KiNativ -- single dose experiment - Dataset (ID:20103)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| XMD-12 | PC-3 | M3K2 | ELAVkQVQFDPDSPETSKEVNALECEIQLLK | Lys1 | 75.4 | 10 | uM |
| XMD-12 | PC-3 | PKD2 | DVAVkVIDK | Lys1 | 33.2 | 10 | uM |
| XMD-12 | PC-3 | M3K2,MAP3K3 | DIkGANILR | Lys2 | 18.0 | 10 | uM |
| XMD-12 | PC-3 | MLTK | WISQDKEVAVKk | Lys1 | 15.8 | 10 | uM |
| XMD-12 | PC-3 | MAP3K4 | DIkGANIFLTSSGLIK | Lys2 | -0.6 | 10 | uM |
| XMD-12 | PC-3 | EGFR | LLGAEEKEYHAEGGkVPIK | Activation Loop | -26.4 | 10 | uM |
| XMD-12 | PC-3 | ZC1/HGK,ZC2/TNIK,ZC3/MINK | DIkGQNVLLTENAEVK | Lys2 | -7.1 | 10 | uM |
| XMD-12 | PC-3 | MARK2,MARK3 | DLkAENLLLDADMNIK | Lys2 | 72.5 | 10 | uM |
| XMD-12 | PC-3 | CLK2 | LTHTDLkPENILFVNSDYELTYNLEK | Lys2 | 5.8 | 10 | uM |
| XMD-12 | PC-3 | PRP4 | CNILHADIkPDNILVNESK | Lys2 | -13.9 | 10 | uM |
| XMD-12 | PC-3 | MAST3 | DLkPDNLLITSLGHIK | Lys2 | 15.2 | 10 | uM |
| XMD-12 | PC-3 | ANPb | GMAFLHNSIISSHGSLkSSNCVVDSR | Lys2 | -7.0 | 10 | uM |
| XMD-12 | PC-3 | MLK3 | DLkSNNILLLQPIESDDMEHK | Lys2 | 40.1 | 10 | uM |
| XMD-12 | PC-3 | CDK5 | DLkPQNLLINR | Lys2 | 12.5 | 10 | uM |
| XMD-12 | PC-3 | MPSK1 | DLkPTNILLGDEGQPVLMDLGSMNQACIHVEGSR | Lys2 | 81.1 | 10 | uM |
| XMD-12 | PC-3 | CaMK2a,CaMK2b,CaMK2d,CaMK2g | DLkPENLLLASK | Lys2 | 23.5 | 10 | uM |
| XMD-12 | PC-3 | CDK5 | ETHEIVALkR | Lys1 | 4.5 | 10 | uM |
| XMD-12 | PC-3 | CHK2 | DLkPENVLLSSQEEDCLIK | Lys2 | 29.7 | 10 | uM |
| XMD-12 | PC-3 | MST1 | ETGQIVAIkQVPVESDLQEIIK | Lys1 | 73.5 | 10 | uM |
| XMD-12 | PC-3 | MST1,MST2 | DIkAGNILLNTEGHAK | Lys2 | 39.1 | 10 | uM |
| XMD-12 | PC-3 | CK2a2 | DVkPHNVMIDHQQK | Lys2 | 33.4 | 10 | uM |
| XMD-12 | PC-3 | MST2 | ESGQVVAIkQVPVESDLQEIIK | Lys1 | 53.0 | 10 | uM |
| XMD-12 | PC-3 | EPHB4 | FLEENSSDPTYTSSLGGkIPIR | Activation Loop | 51.7 | 10 | uM |
| XMD-12 | PC-3 | MST4,YSK1 | DIkAANVLLSEQGDVK | Lys2 | 28.6 | 10 | uM |
| XMD-12 | PC-3 | NDR2 | DTGHIYAMkILR | Lys1 | 36.3 | 10 | uM |