XMD-12 KiNativ -- single dose experiment - Dataset (ID:20103)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD-12 PC-3 EGFR
ITDFGLAkLLGAEEK
Activation Loop
-24.0
10
uM
XMD-12 PC-3 EphA1
LLDDFDGTYETQGGkIPIR
Activation Loop
46.7
10
uM
XMD-12 PC-3 NEK6,NEK7
DIkPANVFITATGVVK
Lys2
-24.3
10
uM
XMD-12 PC-3 NEK8
DLkTQNILLDK
Lys2
-31.6
10
uM
XMD-12 PC-3 EPHA2
EVPVAIkTLK
Lys1
8.4
10
uM
XMD-12 PC-3 NEK9
DIkTLNIFLTK
Lys2
-26.4
10
uM
XMD-12 PC-3 EphA7
VIEDDPEAVYTTTGGkIPVR
Activation Loop
-21.4
10
uM
XMD-12 PC-3 NEK9
LGDYGLAkK
Activation Loop
3.4
10
uM
XMD-12 PC-3 EPHB2
FLEDDTSDPTYTSALGGkIPIR
Activation Loop
27.3
10
uM
XMD-12 PC-3 p38d,p38g
DLkPGNLAVNEDCELK
Lys2
-10.2
10
uM
XMD-12 PC-3 TLK1
YAAVkIHQLNK
Lys1
-47.5
10
uM
XMD-12 PC-3 KS6B1
DLkPENIMLNHQGHVK
Lys2
14.0
10
uM
XMD-12 PC-3 p70S6K,p70S6Kb
GGYGkVFQVR
ATP Loop
-1.6
10
uM
XMD-12 PC-3 M3K2
VYLCYDVDTGRELAVkQVQFDPDSPETSKEVNALECEIQLLK
Lys1
66.5
10
uM
XMD-12 PC-3 CDK16
LTDNLVALkEIR
Lys1
-11.1
10
uM
XMD-12 PC-3 GCN2
LDGCCYAVkR
Lys1
-12.4
10
uM